FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB Docking_panel_21Explorer results are being read from this database.
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3 compounds in matrix 6 best compound-target hits listed 6 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T02T03T04T09T12T16
Z27116094
[H]N(CCN1C(=O)S/C(=C/c2cccnc2)C1=O)C(=O)[C@H]1CC(=O)N(c2cccc(SC)c2)C1
0.859 0.854 2 0.86 0.85
Z27116094
[H]N(CCN1C(=O)S/C(=C\c2cccnc2)C1=O)C(=O)[C@@H]1CC(=O)N(c2cccc(SC)c2)C1
0.830 0.804 2 0.83 0.78
Z27116094
[H]N(CCN1C(=O)S/C(=C\c2cccnc2)C1=O)C(=O)[C@H]1CC(=O)N(c2cccc(SC)c2)C1
0.802 0.790 2 0.80 0.78

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
Z27116094
[H]N(CCN1C(=O)S/C(=C/c2cccnc2)C1=O)C(=O)[C@H]1CC(=O)N(c2cccc(SC)c2)C1
T03
native IFP available
T03
dockmulti_91311c650f2e_T03
0.859 1.000 0.597 native_similarity final_rank_score -25.5601 -0.879258 20 1 Pose
Z27116094
[H]N(CCN1C(=O)S/C(=C/c2cccnc2)C1=O)C(=O)[C@H]1CC(=O)N(c2cccc(SC)c2)C1
T12
native IFP available
T12
dockmulti_91311c650f2e_T12
0.849 1.000 0.568 native_similarity final_rank_score -26.9468 -0.669663 15 6 Pose
Z27116094
[H]N(CCN1C(=O)S/C(=C\c2cccnc2)C1=O)C(=O)[C@@H]1CC(=O)N(c2cccc(SC)c2)C1
T02
native IFP available
T02
dockmulti_91311c650f2e_T02
0.830 1.000 0.515 native_similarity final_rank_score -29.5722 -0.757948 21 1 Pose
Z27116094
[H]N(CCN1C(=O)S/C(=C\c2cccnc2)C1=O)C(=O)[C@H]1CC(=O)N(c2cccc(SC)c2)C1
T09
native IFP available
T09
dockmulti_91311c650f2e_T09
0.802 1.000 0.433 native_similarity final_rank_score -25.0882 -0.716024 17 2 Pose
Z27116094
[H]N(CCN1C(=O)S/C(=C\c2cccnc2)C1=O)C(=O)[C@H]1CC(=O)N(c2cccc(SC)c2)C1
T16
native IFP available
T16
dockmulti_91311c650f2e_T16
0.779 1.000 0.368 native_similarity final_rank_score -24.6649 -0.607112 15 3 Pose
Z27116094
[H]N(CCN1C(=O)S/C(=C\c2cccnc2)C1=O)C(=O)[C@@H]1CC(=O)N(c2cccc(SC)c2)C1
T04
native IFP available
T04
dockmulti_91311c650f2e_T04
0.778 1.000 0.365 native_similarity final_rank_score -22.0526 -0.571642 15 1 Pose