FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB fairmolExplorer results are being read from this database.
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6 compounds in matrix 12 best compound-target hits listed 11 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T01T02T03T06T09T10T12T16T18T21T22
Z104500108
[H]Oc1ccc(/C=C\C(=O)CC(=O)/C=C\c2ccc(O)c(OC)c2)cc1OC
0.941 0.865 2 0.94 0.79
Z104500108
[H]Oc1ccc(/C=C\C(O)=C\C(=O)/C=C/c2ccc(O[H])c(OC)c2)cc1OC
0.927 0.899 3 0.86 0.91 0.93
Z104500108
[H]Oc1ccc(/C=C\C(=O)CC(=O)/C=C/c2ccc(O[H])c(OC)c2)cc1OC
0.913 0.912 2 0.91 0.91
Z104500108
[H]Oc1ccc(/C=C/C(=O)/C=C(O)/C=C/c2ccc(O[H])c(OC)c2)cc1OC
0.913 0.863 3 0.84 0.84 0.91
Z104500108
[H]OC(=C\C(=O)/C=C\c1ccc(O[H])c(OC)c1)/C=C/c1ccc(O[H])c(OC)c1
0.838 0.838 1 0.84
Z104500108
[H]Oc1ccc(/C=C\C(=O)/C=C(O)/C=C\c2ccc(O[H])c(OC)c2)cc1OC
0.743 0.743 1 0.74

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
Z104500108
[H]Oc1ccc(/C=C\C(=O)CC(=O)/C=C\c2ccc(O)c(OC)c2)cc1OC
T10
native IFP available
T10
selection_import_t10
0.941 1.000 0.832 native_similarity final_rank_score -18.9139 -0.939358 18 11 Pose
Z104500108
[H]Oc1ccc(/C=C\C(O)=C\C(=O)/C=C/c2ccc(O[H])c(OC)c2)cc1OC
T22
native IFP available
T22
selection_import_t22
0.927 1.000 0.792 native_similarity final_rank_score -24.004 -1.15571 23 12 Pose
Z104500108
[H]Oc1ccc(/C=C\C(=O)CC(=O)/C=C/c2ccc(O[H])c(OC)c2)cc1OC
T03
native IFP available
T03
selection_import_t03
0.913 1.000 0.751 native_similarity final_rank_score -24.4552 -1.0097 16 6 Pose
Z104500108
[H]Oc1ccc(/C=C/C(=O)/C=C(O)/C=C/c2ccc(O[H])c(OC)c2)cc1OC
T21
native IFP available
T21
selection_import_t21
0.913 1.000 0.750 native_similarity final_rank_score -15.4446 -0.91695 18 9 Pose
Z104500108
[H]Oc1ccc(/C=C\C(=O)CC(=O)/C=C/c2ccc(O[H])c(OC)c2)cc1OC
T21
native IFP available
T21
selection_import_t21
0.911 1.000 0.746 native_similarity final_rank_score -18.0333 -0.928261 16 13 Pose
Z104500108
[H]Oc1ccc(/C=C\C(O)=C\C(=O)/C=C/c2ccc(O[H])c(OC)c2)cc1OC
T12
native IFP available
T12
selection_import_t12
0.906 1.000 0.731 native_similarity final_rank_score -18.7671 -1.02624 19 10 Pose
Z104500108
[H]Oc1ccc(/C=C\C(O)=C\C(=O)/C=C/c2ccc(O[H])c(OC)c2)cc1OC
T06
native IFP available
T06
selection_import_t06
0.865 1.000 0.614 native_similarity final_rank_score -18.2139 -0.97482 18 3 Pose
Z104500108
[H]Oc1ccc(/C=C/C(=O)/C=C(O)/C=C/c2ccc(O[H])c(OC)c2)cc1OC
T01
native IFP available
T01
selection_import_t01
0.838 1.000 0.536 native_similarity final_rank_score -24.155 -0.947352 17 6 Pose
Z104500108
[H]Oc1ccc(/C=C/C(=O)/C=C(O)/C=C/c2ccc(O[H])c(OC)c2)cc1OC
T02
native IFP available
T02
selection_import_t02
0.838 1.000 0.536 native_similarity final_rank_score -23.6282 -0.940821 17 6 Pose
Z104500108
[H]OC(=C\C(=O)/C=C\c1ccc(O[H])c(OC)c1)/C=C/c1ccc(O[H])c(OC)c1
T09
native IFP available
T09
selection_import_t09
0.838 1.000 0.536 native_similarity final_rank_score -26.8366 -0.952526 18 9 Pose
Z104500108
[H]Oc1ccc(/C=C\C(=O)CC(=O)/C=C\c2ccc(O)c(OC)c2)cc1OC
T18
native IFP available
T18
selection_import_t18
0.789 1.000 0.397 native_similarity final_rank_score -24.3432 -0.945628 15 5 Pose
Z104500108
[H]Oc1ccc(/C=C\C(=O)/C=C(O)/C=C\c2ccc(O[H])c(OC)c2)cc1OC
T16
native IFP available
T16
selection_import_t16
0.743 1.000 0.264 native_similarity final_rank_score -17.8909 -0.858455 15 8 Pose