FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB fairmolExplorer results are being read from this database.
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3 compounds in matrix 3 best compound-target hits listed 3 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T01T12T21
TC107
[H]Oc1ccc2c(c1)CC[C@@H]1[C@@H]2CC[C@]2(C)c3nn(CCOC)cc3C[C@@H]12
0.907 0.907 1 0.91
TC107
[H]Oc1ccc2c(c1)CC[C@H]1[C@H]2CC[C@]2(C)c3c(cn(CCOC)[n+]3[H])C[C@@H]12
0.902 0.902 1 0.90
TC107
[H]Oc1ccc2c(c1)CC[C@H]1[C@H]3Cc4cn(CCOC)[n+]([H])c4[C@@]3(C)CC[C@@H]21
0.869 0.869 1 0.87

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
TC107
[H]Oc1ccc2c(c1)CC[C@@H]1[C@@H]2CC[C@]2(C)c3nn(CCOC)cc3C[C@@H]12
T12
native IFP available
T12
selection_import_t12
0.907 1.000 0.736 native_similarity final_rank_score -28.5316 -1.0982 18 6 Pose
TC107
[H]Oc1ccc2c(c1)CC[C@H]1[C@H]2CC[C@]2(C)c3c(cn(CCOC)[n+]3[H])C[C@@H]12
T21
native IFP available
T21
selection_import_t21
0.902 1.000 0.720 native_similarity final_rank_score -24.3297 -1.01378 15 6 Pose
TC107
[H]Oc1ccc2c(c1)CC[C@H]1[C@H]3Cc4cn(CCOC)[n+]([H])c4[C@@]3(C)CC[C@@H]21
T01
native IFP available
T01
selection_import_t01
0.869 1.000 0.627 native_similarity final_rank_score -25.2322 -1.00797 17 3 Pose