FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB Docking_panel_21Explorer results are being read from this database.
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2 compounds in matrix 5 best compound-target hits listed 5 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T03T15T16T18T20
OSA_Lib_70
[H][N+]([H])([H])CCN1CC[C@]2([N+]3([H])CCCCC3)C[C@@H](c3ccc(Cl)cc3)[C@H]1[C@H](c1ccc(Cl)cc1)C2
0.962 0.842 4 0.84 0.80 0.76 0.96
OSA_Lib_70
[H][N+]([H])([H])CCN1CC[C@]2([N+]3([H])CCCCC3)C[C@H](c3ccc(Cl)cc3)[C@H]1[C@@H](c1ccc(Cl)cc1)C2
0.789 0.789 1 0.79

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
OSA_Lib_70
[H][N+]([H])([H])CCN1CC[C@]2([N+]3([H])CCCCC3)C[C@@H](c3ccc(Cl)cc3)[C@H]1[C@H](c1ccc(Cl)cc1)C2
T20
native IFP available
T20
dockmulti_91311c650f2e_T20
0.962 1.000 0.891 native_similarity final_rank_score -14.556 -0.464422 11 2 Pose
OSA_Lib_70
[H][N+]([H])([H])CCN1CC[C@]2([N+]3([H])CCCCC3)C[C@@H](c3ccc(Cl)cc3)[C@H]1[C@H](c1ccc(Cl)cc1)C2
T03
native IFP available
T03
dockmulti_91311c650f2e_T03
0.843 1.000 0.551 native_similarity final_rank_score -24.2002 -0.775874 20 0 Pose
OSA_Lib_70
[H][N+]([H])([H])CCN1CC[C@]2([N+]3([H])CCCCC3)C[C@@H](c3ccc(Cl)cc3)[C@H]1[C@H](c1ccc(Cl)cc1)C2
T16
native IFP available
T16
dockmulti_91311c650f2e_T16
0.800 0.970 0.485 native_similarity final_rank_score -17.2604 -0.696198 15 3 Pose
OSA_Lib_70
[H][N+]([H])([H])CCN1CC[C@]2([N+]3([H])CCCCC3)C[C@H](c3ccc(Cl)cc3)[C@H]1[C@@H](c1ccc(Cl)cc1)C2
T15
native IFP available
T15
dockmulti_91311c650f2e_T15
0.789 1.000 0.397 native_similarity final_rank_score -21.212 -0.710495 15 2 Pose
OSA_Lib_70
[H][N+]([H])([H])CCN1CC[C@]2([N+]3([H])CCCCC3)C[C@@H](c3ccc(Cl)cc3)[C@H]1[C@H](c1ccc(Cl)cc1)C2
T18
native IFP available
T18
dockmulti_91311c650f2e_T18
0.764 1.000 0.326 native_similarity final_rank_score -14.6552 -0.528601 11 1 Pose