FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB SELECTIONExplorer results are being read from this database.
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2 compounds in matrix 3 best compound-target hits listed 3 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T01T03T15
OSA_Lib_305
[H][N@@+]1(Cc2ccncc2)C[C@H]2[C@@H](c3ccccc3)C[C@](N3CCCC3)(C[C@H]2c2ccccc2)C1
0.844 0.844 1 0.84
OSA_Lib_305
[H][N@@+]1(Cc2ccncc2)C[C@H]2[C@@H](c3ccccc3)C[C@](N3CCCC3)(C[C@@H]2c2ccccc2)C1
0.827 0.818 2 0.83 0.81

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
OSA_Lib_305
[H][N@@+]1(Cc2ccncc2)C[C@H]2[C@@H](c3ccccc3)C[C@](N3CCCC3)(C[C@H]2c2ccccc2)C1
T01
native IFP available
T01
selection_import_t01
0.844 1.000 0.555 native_similarity final_rank_score -23.182 -0.783524 19 1 Pose
OSA_Lib_305
[H][N@@+]1(Cc2ccncc2)C[C@H]2[C@@H](c3ccccc3)C[C@](N3CCCC3)(C[C@@H]2c2ccccc2)C1
T03
native IFP available
T03
selection_import_t03
0.827 1.000 0.507 native_similarity final_rank_score -26.8159 -0.822958 20 1 Pose
OSA_Lib_305
[H][N@@+]1(Cc2ccncc2)C[C@H]2[C@@H](c3ccccc3)C[C@](N3CCCC3)(C[C@@H]2c2ccccc2)C1
T15
native IFP available
T15
selection_import_t15
0.809 1.000 0.453 native_similarity final_rank_score -24.6348 -0.742144 15 2 Pose