FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB Docking_panel_21Explorer results are being read from this database.
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4 compounds in matrix 4 best compound-target hits listed 4 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T03T15T16T20
OSA_Lib_240
[H]N(C(=O)C[N+]1([H])CCCC1)[C@H]1C[C@]2([N+]3([H])CCCCC3)C[C@@H](c3ccccc3)[C@H]1[C@H](c1ccccc1)C2
0.894 0.894 1 0.89
OSA_Lib_240
[H]N(C(=O)CN1CCCC1)[C@H]1C[C@]2([N+]3([H])CCCCC3)C[C@H](c3ccccc3)[C@H]1[C@@H](c1ccccc1)C2
0.827 0.827 1 0.83
OSA_Lib_240
[H]N(C(=O)C[N+]1([H])CCCC1)[C@H]1C[C@]2([N+]3([H])CCCCC3)C[C@H](c3ccccc3)[C@H]1[C@H](c1ccccc1)C2
0.825 0.825 1 0.82
OSA_Lib_240
[H]N(C(=O)C[N+]1([H])CCCC1)[C@@H]1C[C@]2([N+]3([H])CCCCC3)C[C@@H](c3ccccc3)[C@H]1[C@H](c1ccccc1)C2
0.817 0.817 1 0.82

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
OSA_Lib_240
[H]N(C(=O)C[N+]1([H])CCCC1)[C@H]1C[C@]2([N+]3([H])CCCCC3)C[C@@H](c3ccccc3)[C@H]1[C@H](c1ccccc1)C2
T20
native IFP available
T20
dockmulti_91311c650f2e_T20
0.894 1.000 0.696 native_similarity final_rank_score -19.9518 -0.493841 12 4 Pose
OSA_Lib_240
[H]N(C(=O)CN1CCCC1)[C@H]1C[C@]2([N+]3([H])CCCCC3)C[C@H](c3ccccc3)[C@H]1[C@@H](c1ccccc1)C2
T03
native IFP available
T03
dockmulti_91311c650f2e_T03
0.827 1.000 0.507 native_similarity final_rank_score -24.5515 -0.725624 20 0 Pose
OSA_Lib_240
[H]N(C(=O)C[N+]1([H])CCCC1)[C@H]1C[C@]2([N+]3([H])CCCCC3)C[C@H](c3ccccc3)[C@H]1[C@H](c1ccccc1)C2
T16
native IFP available
T16
dockmulti_91311c650f2e_T16
0.825 1.000 0.500 native_similarity final_rank_score -21.9917 -0.589155 14 1 Pose
OSA_Lib_240
[H]N(C(=O)C[N+]1([H])CCCC1)[C@@H]1C[C@]2([N+]3([H])CCCCC3)C[C@@H](c3ccccc3)[C@H]1[C@H](c1ccccc1)C2
T15
native IFP available
T15
dockmulti_91311c650f2e_T15
0.817 0.988 0.498 native_similarity final_rank_score -15.0245 -0.451812 16 1 Pose