FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB Docking_panel_21Explorer results are being read from this database.
Reset
3 compounds in matrix 3 best compound-target hits listed 3 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T03T15T16
OSA_Lib_239
[H][N+]([H])(CN1CCCC1)[C@@H]1C[C@]2([N+]([H])(C)C)C[C@@H](c3ccccc3)[C@H]1[C@H](c1ccccc1)C2
0.854 0.854 1 0.85
OSA_Lib_239
[H]N(C[N+]1([H])CCCC1)[C@@H]1C[C@]2([N+]([H])(C)C)C[C@H](c3ccccc3)[C@H]1[C@@H](c1ccccc1)C2
0.809 0.809 1 0.81
OSA_Lib_239
[H]N(C[N+]1([H])CCCC1)[C@H]1C[C@@]2([N+]([H])(C)C)C[C@H](c3ccccc3)[C@@H]1[C@H](c1ccccc1)C2
0.781 0.781 1 0.78

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
OSA_Lib_239
[H][N+]([H])(CN1CCCC1)[C@@H]1C[C@]2([N+]([H])(C)C)C[C@@H](c3ccccc3)[C@H]1[C@H](c1ccccc1)C2
T03
native IFP available
T03
dockmulti_91311c650f2e_T03
0.854 1.000 0.583 native_similarity final_rank_score -25.7538 -0.858111 21 0 Pose
OSA_Lib_239
[H]N(C[N+]1([H])CCCC1)[C@@H]1C[C@]2([N+]([H])(C)C)C[C@H](c3ccccc3)[C@H]1[C@@H](c1ccccc1)C2
T15
native IFP available
T15
dockmulti_91311c650f2e_T15
0.809 1.000 0.453 native_similarity final_rank_score -21.1762 -0.636541 15 1 Pose
OSA_Lib_239
[H]N(C[N+]1([H])CCCC1)[C@H]1C[C@@]2([N+]([H])(C)C)C[C@H](c3ccccc3)[C@@H]1[C@H](c1ccccc1)C2
T16
native IFP available
T16
dockmulti_91311c650f2e_T16
0.781 0.967 0.437 native_similarity final_rank_score -18.6735 -0.580089 14 3 Pose