FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB Docking_panel_21Explorer results are being read from this database.
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3 compounds in matrix 4 best compound-target hits listed 4 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T02T03T10T21
OSA_Lib_109
[H][N+]1([C@]23C[C@H](OC(=O)c4ccc5c(c4)OCO5)[C@H]([C@H](c4ccccc4)C2)[C@H](c2ccccc2)C3)CCCC1
0.922 0.900 2 0.88 0.92
OSA_Lib_109
[H][N+]1([C@]23C[C@H](c4ccccc4)[C@H]([C@H](OC(=O)c4ccc5c(c4)OCO5)C2)[C@H](c2ccccc2)C3)CCCC1
0.841 0.841 1 0.84
OSA_Lib_109
[H][N+]1([C@@]23C[C@H](c4ccccc4)[C@@H]([C@H](OC(=O)c4ccc5c(c4)OCO5)C2)[C@H](c2ccccc2)C3)CCCC1
0.812 0.812 1 0.81

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
OSA_Lib_109
[H][N+]1([C@]23C[C@H](OC(=O)c4ccc5c(c4)OCO5)[C@H]([C@H](c4ccccc4)C2)[C@H](c2ccccc2)C3)CCCC1
T21
native IFP available
T21
dockmulti_91311c650f2e_T21
0.922 1.000 0.777 native_similarity final_rank_score -20.731 -0.5725 15 5 Pose
OSA_Lib_109
[H][N+]1([C@]23C[C@H](OC(=O)c4ccc5c(c4)OCO5)[C@H]([C@H](c4ccccc4)C2)[C@H](c2ccccc2)C3)CCCC1
T10
native IFP available
T10
dockmulti_91311c650f2e_T10
0.879 1.000 0.653 native_similarity final_rank_score -13.4213 -0.601537 13 7 Pose
OSA_Lib_109
[H][N+]1([C@]23C[C@H](c4ccccc4)[C@H]([C@H](OC(=O)c4ccc5c(c4)OCO5)C2)[C@H](c2ccccc2)C3)CCCC1
T03
native IFP available
T03
dockmulti_91311c650f2e_T03
0.841 1.000 0.545 native_similarity final_rank_score -18.6413 -0.602657 17 3 Pose
OSA_Lib_109
[H][N+]1([C@@]23C[C@H](c4ccccc4)[C@@H]([C@H](OC(=O)c4ccc5c(c4)OCO5)C2)[C@H](c2ccccc2)C3)CCCC1
T02
native IFP available
T02
dockmulti_91311c650f2e_T02
0.812 1.000 0.464 native_similarity final_rank_score -17.6835 -0.701477 18 1 Pose