FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB fairmolExplorer results are being read from this database.
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1 compounds in matrix 14 best compound-target hits listed 14 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T01T02T05T06T08T09T10T12T14T16T17T18T19T21
OHD_Schistosoma_119
[H]ON([H])C(=O)/C=C/c1ccccc1CSc1nc(Cc2ccccc2)cc(=O)n1[H]
0.915 0.834 14 0.81 0.81 0.85 0.91 0.85 0.81 0.89 0.88 0.85 0.77 0.81 0.79 0.75 0.92

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
OHD_Schistosoma_119
[H]ON([H])C(=O)/C=C/c1ccccc1CSc1nc(Cc2ccccc2)cc(=O)n1[H]
T21
native IFP available
T21
selection_import_t21
0.915 1.000 0.758 native_similarity final_rank_score -29.9241 -1.08027 16 11 Pose
OHD_Schistosoma_119
[H]ON([H])C(=O)/C=C/c1ccccc1CSc1nc(Cc2ccccc2)cc(=O)n1[H]
T06
native IFP available
T06
selection_import_t06
0.913 1.000 0.751 native_similarity final_rank_score -25.8329 -0.94766 20 7 Pose
OHD_Schistosoma_119
[H]ON([H])C(=O)/C=C/c1ccccc1CSc1nc(Cc2ccccc2)cc(=O)n1[H]
T10
native IFP available
T10
selection_import_t10
0.886 1.000 0.674 native_similarity final_rank_score -28.4656 -0.958338 18 9 Pose
OHD_Schistosoma_119
[H]ON([H])C(=O)/C=C/c1ccccc1CSc1nc(Cc2ccccc2)cc(=O)n1[H]
T12
native IFP available
T12
selection_import_t12
0.884 1.000 0.667 native_similarity final_rank_score -27.9224 -1.13445 16 13 Pose
OHD_Schistosoma_119
[H]ON([H])C(=O)/C=C/c1ccccc1CSc1nc(Cc2ccccc2)cc(=O)n1[H]
T08
native IFP available
T08
selection_import_t08
0.851 1.000 0.573 native_similarity final_rank_score -31.1202 -1.15406 15 9 Pose
OHD_Schistosoma_119
[H]ON([H])C(=O)/C=C/c1ccccc1CSc1nc(Cc2ccccc2)cc(=O)n1[H]
T05
native IFP available
T05
selection_import_t05
0.847 1.000 0.564 native_similarity final_rank_score -32.9082 -1.06988 15 7 Pose
OHD_Schistosoma_119
[H]ON([H])C(=O)/C=C/c1ccccc1CSc1nc(Cc2ccccc2)cc(=O)n1[H]
T14
native IFP available
T14
selection_import_t14
0.846 1.000 0.560 native_similarity final_rank_score -23.1448 -0.880375 16 9 Pose
OHD_Schistosoma_119
[H]ON([H])C(=O)/C=C/c1ccccc1CSc1nc(Cc2ccccc2)cc(=O)n1[H]
T01
native IFP available
T01
selection_import_t01
0.809 1.000 0.454 native_similarity final_rank_score -33.9816 -1.14501 17 4 Pose
OHD_Schistosoma_119
[H]ON([H])C(=O)/C=C/c1ccccc1CSc1nc(Cc2ccccc2)cc(=O)n1[H]
T02
native IFP available
T02
selection_import_t02
0.809 1.000 0.453 native_similarity final_rank_score -24.0652 -0.956091 15 3 Pose
OHD_Schistosoma_119
[H]ON([H])C(=O)/C=C/c1ccccc1CSc1nc(Cc2ccccc2)cc(=O)n1[H]
T09
native IFP available
T09
selection_import_t09
0.808 1.000 0.452 native_similarity final_rank_score -26.0298 -1.03576 16 5 Pose
OHD_Schistosoma_119
[H]ON([H])C(=O)/C=C/c1ccccc1CSc1nc(Cc2ccccc2)cc(=O)n1[H]
T17
native IFP available
T17
selection_import_t17
0.806 1.000 0.445 native_similarity final_rank_score -25.4605 -0.886989 18 8 Pose
OHD_Schistosoma_119
[H]ON([H])C(=O)/C=C/c1ccccc1CSc1nc(Cc2ccccc2)cc(=O)n1[H]
T18
native IFP available
T18
selection_import_t18
0.789 1.000 0.397 native_similarity final_rank_score -22.1294 -0.805172 15 8 Pose
OHD_Schistosoma_119
[H]ON([H])C(=O)/C=C/c1ccccc1CSc1nc(Cc2ccccc2)cc(=O)n1[H]
T16
native IFP available
T16
selection_import_t16
0.766 1.000 0.331 native_similarity final_rank_score -22.4978 -0.820834 13 7 Pose
OHD_Schistosoma_119
[H]ON([H])C(=O)/C=C/c1ccccc1CSc1nc(Cc2ccccc2)cc(=O)n1[H]
T19
native IFP available
T19
selection_import_t19
0.748 1.000 0.280 native_similarity final_rank_score -29.6204 -1.19861 19 13 Pose