FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB fairmolExplorer results are being read from this database.
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2 compounds in matrix 12 best compound-target hits listed 12 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T01T02T08T09T10T12T15T16T18T19T20T21
OHD_MAC_68
[H]Oc1cc(/C=[N+]([H])/N=c2\c3nc[n+]([H])c(N([H])c4ccc(Cl)c(C(F)(F)F)c4)c3ncn2[H])cc(O[H])c1O[H]
0.946 0.921 3 0.90 0.91 0.95
OHD_MAC_68
[H]Oc1cc(/C=N/N([H])c2ncnc3c(N([H])c4ccc(Cl)c(C(F)(F)F)c4)ncnc23)cc(O[H])c1O[H]
0.932 0.832 9 0.87 0.83 0.89 0.93 0.75 0.73 0.82 0.75 0.91

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
OHD_MAC_68
[H]Oc1cc(/C=[N+]([H])/N=c2\c3nc[n+]([H])c(N([H])c4ccc(Cl)c(C(F)(F)F)c4)c3ncn2[H])cc(O[H])c1O[H]
T20
native IFP available
T20
selection_import_t20
0.946 1.000 0.846 native_similarity final_rank_score -17.636 -0.557853 13 9 Pose
OHD_MAC_68
[H]Oc1cc(/C=N/N([H])c2ncnc3c(N([H])c4ccc(Cl)c(C(F)(F)F)c4)ncnc23)cc(O[H])c1O[H]
T12
native IFP available
T12
selection_import_t12
0.932 1.000 0.805 native_similarity final_rank_score -19.8732 -0.875736 17 13 Pose
OHD_MAC_68
[H]Oc1cc(/C=[N+]([H])/N=c2\c3nc[n+]([H])c(N([H])c4ccc(Cl)c(C(F)(F)F)c4)c3ncn2[H])cc(O[H])c1O[H]
T10
native IFP available
T10
selection_import_t10
0.913 1.000 0.751 native_similarity final_rank_score -23.4425 -0.742386 21 9 Pose
OHD_MAC_68
[H]Oc1cc(/C=N/N([H])c2ncnc3c(N([H])c4ccc(Cl)c(C(F)(F)F)c4)ncnc23)cc(O[H])c1O[H]
T21
native IFP available
T21
selection_import_t21
0.911 1.000 0.747 native_similarity final_rank_score -22.2807 -0.781983 19 14 Pose
OHD_MAC_68
[H]Oc1cc(/C=[N+]([H])/N=c2\c3nc[n+]([H])c(N([H])c4ccc(Cl)c(C(F)(F)F)c4)c3ncn2[H])cc(O[H])c1O[H]
T08
native IFP available
T08
selection_import_t08
0.904 1.000 0.727 native_similarity final_rank_score -30.4064 -1.03229 20 9 Pose
OHD_MAC_68
[H]Oc1cc(/C=N/N([H])c2ncnc3c(N([H])c4ccc(Cl)c(C(F)(F)F)c4)ncnc23)cc(O[H])c1O[H]
T09
native IFP available
T09
selection_import_t09
0.889 1.000 0.683 native_similarity final_rank_score -16.7453 -0.774291 19 4 Pose
OHD_MAC_68
[H]Oc1cc(/C=N/N([H])c2ncnc3c(N([H])c4ccc(Cl)c(C(F)(F)F)c4)ncnc23)cc(O[H])c1O[H]
T01
native IFP available
T01
selection_import_t01
0.871 1.000 0.630 native_similarity final_rank_score -22.4146 -0.841884 20 7 Pose
OHD_MAC_68
[H]Oc1cc(/C=N/N([H])c2ncnc3c(N([H])c4ccc(Cl)c(C(F)(F)F)c4)ncnc23)cc(O[H])c1O[H]
T02
native IFP available
T02
selection_import_t02
0.834 1.000 0.524 native_similarity final_rank_score -17.8711 -0.825357 18 8 Pose
OHD_MAC_68
[H]Oc1cc(/C=N/N([H])c2ncnc3c(N([H])c4ccc(Cl)c(C(F)(F)F)c4)ncnc23)cc(O[H])c1O[H]
T18
native IFP available
T18
selection_import_t18
0.820 1.000 0.485 native_similarity final_rank_score -20.9447 -0.692916 17 7 Pose
OHD_MAC_68
[H]Oc1cc(/C=N/N([H])c2ncnc3c(N([H])c4ccc(Cl)c(C(F)(F)F)c4)ncnc23)cc(O[H])c1O[H]
T19
native IFP available
T19
selection_import_t19
0.752 1.000 0.291 native_similarity final_rank_score -22.3139 -0.925959 24 12 Pose
OHD_MAC_68
[H]Oc1cc(/C=N/N([H])c2ncnc3c(N([H])c4ccc(Cl)c(C(F)(F)F)c4)ncnc23)cc(O[H])c1O[H]
T15
native IFP available
T15
selection_import_t15
0.746 1.000 0.274 native_similarity final_rank_score -19.5716 -0.736534 19 5 Pose
OHD_MAC_68
[H]Oc1cc(/C=N/N([H])c2ncnc3c(N([H])c4ccc(Cl)c(C(F)(F)F)c4)ncnc23)cc(O[H])c1O[H]
T16
native IFP available
T16
selection_import_t16
0.731 1.000 0.230 native_similarity final_rank_score -19.8123 -0.697837 12 6 Pose