FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB fairmolExplorer results are being read from this database.
Reset
2 compounds in matrix 8 best compound-target hits listed 8 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T01T02T03T06T07T08T11T14
OHD_Babesia_62
[H]N([H])c1nc2ccc(CN([H])c3cc(OC)ccc3OC)c(Cl)c2c(N([H])[H])[n+]1[H]
0.974 0.876 7 0.87 0.86 0.84 0.97 0.89 0.90 0.80
OHD_Babesia_62
[H]N([H])c1nc(N([H])[H])c2c(Cl)c(CN([H])c3cc(OC)ccc3OC)ccc2n1
0.785 0.785 1 0.78

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
OHD_Babesia_62
[H]N([H])c1nc2ccc(CN([H])c3cc(OC)ccc3OC)c(Cl)c2c(N([H])[H])[n+]1[H]
T06
native IFP available
T06
selection_import_t06
0.974 1.000 0.925 native_similarity final_rank_score -27.1771 -1.13474 21 5 Pose
OHD_Babesia_62
[H]N([H])c1nc2ccc(CN([H])c3cc(OC)ccc3OC)c(Cl)c2c(N([H])[H])[n+]1[H]
T08
native IFP available
T08
selection_import_t08
0.903 1.000 0.724 native_similarity final_rank_score -36.1942 -1.45605 19 6 Pose
OHD_Babesia_62
[H]N([H])c1nc2ccc(CN([H])c3cc(OC)ccc3OC)c(Cl)c2c(N([H])[H])[n+]1[H]
T07
native IFP available
T07
selection_import_t07
0.888 1.000 0.681 native_similarity final_rank_score -37.0939 -1.43855 15 7 Pose
OHD_Babesia_62
[H]N([H])c1nc2ccc(CN([H])c3cc(OC)ccc3OC)c(Cl)c2c(N([H])[H])[n+]1[H]
T01
native IFP available
T01
selection_import_t01
0.866 1.000 0.617 native_similarity final_rank_score -26.1007 -1.03179 21 10 Pose
OHD_Babesia_62
[H]N([H])c1nc2ccc(CN([H])c3cc(OC)ccc3OC)c(Cl)c2c(N([H])[H])[n+]1[H]
T02
native IFP available
T02
selection_import_t02
0.855 1.000 0.586 native_similarity final_rank_score -27.8978 -1.11322 20 9 Pose
OHD_Babesia_62
[H]N([H])c1nc2ccc(CN([H])c3cc(OC)ccc3OC)c(Cl)c2c(N([H])[H])[n+]1[H]
T03
native IFP available
T03
selection_import_t03
0.841 1.000 0.545 native_similarity final_rank_score -29.4478 -1.15696 18 11 Pose
OHD_Babesia_62
[H]N([H])c1nc2ccc(CN([H])c3cc(OC)ccc3OC)c(Cl)c2c(N([H])[H])[n+]1[H]
T14
native IFP available
T14
selection_import_t14
0.804 1.000 0.440 native_similarity final_rank_score -21.8572 -0.910007 13 6 Pose
OHD_Babesia_62
[H]N([H])c1nc(N([H])[H])c2c(Cl)c(CN([H])c3cc(OC)ccc3OC)ccc2n1
T11
native IFP available
T11
selection_import_t11
0.785 1.000 0.385 native_similarity final_rank_score -18.3996 -1.05369 20 9 Pose