FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB fairmolExplorer results are being read from this database.
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1 compounds in matrix 19 best compound-target hits listed 19 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T01T02T03T04T05T06T09T10T11T12T13T14T15T16T18T19T20T21T22
NMT-TY0929
[H]N([H])c1ccccc1S(=O)(=O)N([H])c1c(N([H])[H])n([H])c(SCc2ccccc2)nc1=O
0.894 0.813 19 0.77 0.79 0.86 0.80 0.88 0.81 0.77 0.85 0.81 0.87 0.89 0.76 0.75 0.76 0.76 0.73 0.89 0.86 0.83

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
NMT-TY0929
[H]N([H])c1ccccc1S(=O)(=O)N([H])c1c(N([H])[H])n([H])c(SCc2ccccc2)nc1=O
T20
native IFP available
T20
selection_import_t20
0.894 1.000 0.696 native_similarity final_rank_score -22.7627 -0.795238 12 7 Pose
NMT-TY0929
[H]N([H])c1ccccc1S(=O)(=O)N([H])c1c(N([H])[H])n([H])c(SCc2ccccc2)nc1=O
T13
native IFP available
T13
selection_import_t13
0.893 1.000 0.694 native_similarity final_rank_score -30.5291 -1.0563 17 13 Pose
NMT-TY0929
[H]N([H])c1ccccc1S(=O)(=O)N([H])c1c(N([H])[H])n([H])c(SCc2ccccc2)nc1=O
T05
native IFP available
T05
selection_import_t05
0.878 1.000 0.652 native_similarity final_rank_score -28.5719 -1.03583 12 7 Pose
NMT-TY0929
[H]N([H])c1ccccc1S(=O)(=O)N([H])c1c(N([H])[H])n([H])c(SCc2ccccc2)nc1=O
T12
native IFP available
T12
selection_import_t12
0.870 1.000 0.628 native_similarity final_rank_score -25.6924 -1.16188 15 10 Pose
NMT-TY0929
[H]N([H])c1ccccc1S(=O)(=O)N([H])c1c(N([H])[H])n([H])c(SCc2ccccc2)nc1=O
T21
native IFP available
T21
selection_import_t21
0.863 1.000 0.609 native_similarity final_rank_score -24.9728 -0.997905 15 12 Pose
NMT-TY0929
[H]N([H])c1ccccc1S(=O)(=O)N([H])c1c(N([H])[H])n([H])c(SCc2ccccc2)nc1=O
T03
native IFP available
T03
selection_import_t03
0.857 1.000 0.591 native_similarity final_rank_score -28.0126 -1.10356 18 4 Pose
NMT-TY0929
[H]N([H])c1ccccc1S(=O)(=O)N([H])c1c(N([H])[H])n([H])c(SCc2ccccc2)nc1=O
T10
native IFP available
T10
selection_import_t10
0.851 1.000 0.575 native_similarity final_rank_score -19.6641 -0.937498 12 16 Pose
NMT-TY0929
[H]N([H])c1ccccc1S(=O)(=O)N([H])c1c(N([H])[H])n([H])c(SCc2ccccc2)nc1=O
T22
native IFP available
T22
selection_import_t22
0.828 1.000 0.509 native_similarity final_rank_score -28.5533 -1.17836 21 9 Pose
NMT-TY0929
[H]N([H])c1ccccc1S(=O)(=O)N([H])c1c(N([H])[H])n([H])c(SCc2ccccc2)nc1=O
T11
native IFP available
T11
selection_import_t11
0.807 1.000 0.450 native_similarity final_rank_score -29.4161 -0.986167 20 5 Pose
NMT-TY0929
[H]N([H])c1ccccc1S(=O)(=O)N([H])c1c(N([H])[H])n([H])c(SCc2ccccc2)nc1=O
T06
native IFP available
T06
selection_import_t06
0.805 1.000 0.443 native_similarity final_rank_score -18.7308 -0.906394 16 3 Pose
NMT-TY0929
[H]N([H])c1ccccc1S(=O)(=O)N([H])c1c(N([H])[H])n([H])c(SCc2ccccc2)nc1=O
T04
native IFP available
T04
selection_import_t04
0.800 1.000 0.429 native_similarity final_rank_score -25.6036 -0.978913 13 2 Pose
NMT-TY0929
[H]N([H])c1ccccc1S(=O)(=O)N([H])c1c(N([H])[H])n([H])c(SCc2ccccc2)nc1=O
T02
native IFP available
T02
selection_import_t02
0.788 1.000 0.393 native_similarity final_rank_score -29.6312 -1.04631 15 5 Pose
NMT-TY0929
[H]N([H])c1ccccc1S(=O)(=O)N([H])c1c(N([H])[H])n([H])c(SCc2ccccc2)nc1=O
T01
native IFP available
T01
selection_import_t01
0.775 1.000 0.357 native_similarity final_rank_score -31.1016 -1.12247 15 6 Pose
NMT-TY0929
[H]N([H])c1ccccc1S(=O)(=O)N([H])c1c(N([H])[H])n([H])c(SCc2ccccc2)nc1=O
T09
native IFP available
T09
selection_import_t09
0.771 1.000 0.347 native_similarity final_rank_score -28.9361 -1.13317 15 12 Pose
NMT-TY0929
[H]N([H])c1ccccc1S(=O)(=O)N([H])c1c(N([H])[H])n([H])c(SCc2ccccc2)nc1=O
T14
native IFP available
T14
selection_import_t14
0.761 1.000 0.317 native_similarity final_rank_score -21.1312 -0.859379 16 9 Pose
NMT-TY0929
[H]N([H])c1ccccc1S(=O)(=O)N([H])c1c(N([H])[H])n([H])c(SCc2ccccc2)nc1=O
T16
native IFP available
T16
selection_import_t16
0.758 1.000 0.308 native_similarity final_rank_score -26.8524 -0.909529 16 10 Pose
NMT-TY0929
[H]N([H])c1ccccc1S(=O)(=O)N([H])c1c(N([H])[H])n([H])c(SCc2ccccc2)nc1=O
T18
native IFP available
T18
selection_import_t18
0.756 1.000 0.302 native_similarity final_rank_score -21.6991 -0.849572 14 9 Pose
NMT-TY0929
[H]N([H])c1ccccc1S(=O)(=O)N([H])c1c(N([H])[H])n([H])c(SCc2ccccc2)nc1=O
T15
native IFP available
T15
selection_import_t15
0.753 1.000 0.295 native_similarity final_rank_score -25.8372 -0.89302 15 8 Pose
NMT-TY0929
[H]N([H])c1ccccc1S(=O)(=O)N([H])c1c(N([H])[H])n([H])c(SCc2ccccc2)nc1=O
T19
native IFP available
T19
selection_import_t19
0.732 1.000 0.235 native_similarity final_rank_score -35.8435 -1.239 17 9 Pose