FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB fairmolExplorer results are being read from this database.
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1 compounds in matrix 16 best compound-target hits listed 16 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T01T02T03T04T06T08T09T11T12T13T15T17T18T20T21T22
NMT-TY0920
[H]N([H])c1ccccc1S(=O)(=O)N([H])c1c(N([H])[H])n([H])c(SCCc2ccccc2)nc1=O
0.939 0.842 16 0.80 0.81 0.75 0.83 0.79 0.87 0.80 0.89 0.88 0.88 0.87 0.76 0.81 0.91 0.94 0.90

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
NMT-TY0920
[H]N([H])c1ccccc1S(=O)(=O)N([H])c1c(N([H])[H])n([H])c(SCCc2ccccc2)nc1=O
T21
native IFP available
T21
selection_import_t21
0.939 1.000 0.825 native_similarity final_rank_score -34.1213 -0.961348 17 11 Pose
NMT-TY0920
[H]N([H])c1ccccc1S(=O)(=O)N([H])c1c(N([H])[H])n([H])c(SCCc2ccccc2)nc1=O
T20
native IFP available
T20
selection_import_t20
0.910 1.000 0.743 native_similarity final_rank_score -25.7042 -0.681525 9 8 Pose
NMT-TY0920
[H]N([H])c1ccccc1S(=O)(=O)N([H])c1c(N([H])[H])n([H])c(SCCc2ccccc2)nc1=O
T22
native IFP available
T22
selection_import_t22
0.895 1.000 0.700 native_similarity final_rank_score -30.3675 -1.24397 26 11 Pose
NMT-TY0920
[H]N([H])c1ccccc1S(=O)(=O)N([H])c1c(N([H])[H])n([H])c(SCCc2ccccc2)nc1=O
T11
native IFP available
T11
selection_import_t11
0.886 1.000 0.676 native_similarity final_rank_score -25.3008 -0.944043 13 5 Pose
NMT-TY0920
[H]N([H])c1ccccc1S(=O)(=O)N([H])c1c(N([H])[H])n([H])c(SCCc2ccccc2)nc1=O
T12
native IFP available
T12
selection_import_t12
0.884 1.000 0.667 native_similarity final_rank_score -35.0271 -1.10054 16 11 Pose
NMT-TY0920
[H]N([H])c1ccccc1S(=O)(=O)N([H])c1c(N([H])[H])n([H])c(SCCc2ccccc2)nc1=O
T13
native IFP available
T13
selection_import_t13
0.876 1.000 0.647 native_similarity final_rank_score -32.0097 -0.981468 17 7 Pose
NMT-TY0920
[H]N([H])c1ccccc1S(=O)(=O)N([H])c1c(N([H])[H])n([H])c(SCCc2ccccc2)nc1=O
T15
native IFP available
T15
selection_import_t15
0.867 1.000 0.620 native_similarity final_rank_score -27.4849 -0.937716 13 10 Pose
NMT-TY0920
[H]N([H])c1ccccc1S(=O)(=O)N([H])c1c(N([H])[H])n([H])c(SCCc2ccccc2)nc1=O
T08
native IFP available
T08
selection_import_t08
0.867 1.000 0.619 native_similarity final_rank_score -30.604 -1.18433 13 9 Pose
NMT-TY0920
[H]N([H])c1ccccc1S(=O)(=O)N([H])c1c(N([H])[H])n([H])c(SCCc2ccccc2)nc1=O
T04
native IFP available
T04
selection_import_t04
0.830 1.000 0.513 native_similarity final_rank_score -23.1229 -0.877657 15 3 Pose
NMT-TY0920
[H]N([H])c1ccccc1S(=O)(=O)N([H])c1c(N([H])[H])n([H])c(SCCc2ccccc2)nc1=O
T02
native IFP available
T02
selection_import_t02
0.811 1.000 0.460 native_similarity final_rank_score -25.1037 -0.935163 14 6 Pose
NMT-TY0920
[H]N([H])c1ccccc1S(=O)(=O)N([H])c1c(N([H])[H])n([H])c(SCCc2ccccc2)nc1=O
T18
native IFP available
T18
selection_import_t18
0.809 1.000 0.453 native_similarity final_rank_score -22.7794 -0.785111 15 9 Pose
NMT-TY0920
[H]N([H])c1ccccc1S(=O)(=O)N([H])c1c(N([H])[H])n([H])c(SCCc2ccccc2)nc1=O
T09
native IFP available
T09
selection_import_t09
0.798 1.000 0.424 native_similarity final_rank_score -28.0195 -0.945999 18 7 Pose
NMT-TY0920
[H]N([H])c1ccccc1S(=O)(=O)N([H])c1c(N([H])[H])n([H])c(SCCc2ccccc2)nc1=O
T01
native IFP available
T01
selection_import_t01
0.798 1.000 0.423 native_similarity final_rank_score -35.0482 -1.01979 16 6 Pose
NMT-TY0920
[H]N([H])c1ccccc1S(=O)(=O)N([H])c1c(N([H])[H])n([H])c(SCCc2ccccc2)nc1=O
T06
native IFP available
T06
selection_import_t06
0.791 1.000 0.402 native_similarity final_rank_score -31.4505 -0.878088 16 3 Pose
NMT-TY0920
[H]N([H])c1ccccc1S(=O)(=O)N([H])c1c(N([H])[H])n([H])c(SCCc2ccccc2)nc1=O
T17
native IFP available
T17
selection_import_t17
0.758 1.000 0.308 native_similarity final_rank_score -33.3801 -0.899682 16 11 Pose
NMT-TY0920
[H]N([H])c1ccccc1S(=O)(=O)N([H])c1c(N([H])[H])n([H])c(SCCc2ccccc2)nc1=O
T03
native IFP available
T03
selection_import_t03
0.754 1.000 0.299 native_similarity final_rank_score -32.8619 -1.04252 15 6 Pose