FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB Docking_panel_21Explorer results are being read from this database.
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2 compounds in matrix 8 best compound-target hits listed 8 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T03T04T06T07T08T09T15T16
NMT-TY0566
[H]N([H])c1ccc(S(=O)(=O)Nc2c[n+]([H])c(N([H])[H])nc2N([H])[H])cc1
0.937 0.928 2 0.94 0.92
NMT-TY0566
[H]N([H])c1ccc(S(=O)(=O)N([H])c2cnc(N([H])[H])nc2N([H])[H])cc1
0.913 0.851 6 0.84 0.90 0.88 0.91 0.80 0.76

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
NMT-TY0566
[H]N([H])c1ccc(S(=O)(=O)Nc2c[n+]([H])c(N([H])[H])nc2N([H])[H])cc1
T06
native IFP available
T06
dockmulti_91311c650f2e_T06
0.937 1.000 0.819 native_similarity final_rank_score -21.3601 -1.23722 17 9 Pose
NMT-TY0566
[H]N([H])c1ccc(S(=O)(=O)Nc2c[n+]([H])c(N([H])[H])nc2N([H])[H])cc1
T08
native IFP available
T08
dockmulti_91311c650f2e_T08
0.919 1.000 0.769 native_similarity final_rank_score -29.8595 -1.65176 16 7 Pose
NMT-TY0566
[H]N([H])c1ccc(S(=O)(=O)N([H])c2cnc(N([H])[H])nc2N([H])[H])cc1
T09
native IFP available
T09
dockmulti_91311c650f2e_T09
0.913 1.000 0.752 native_similarity final_rank_score -24.7621 -1.35166 18 11 Pose
NMT-TY0566
[H]N([H])c1ccc(S(=O)(=O)N([H])c2cnc(N([H])[H])nc2N([H])[H])cc1
T04
native IFP available
T04
dockmulti_91311c650f2e_T04
0.902 1.000 0.719 native_similarity final_rank_score -25.1999 -1.4099 13 5 Pose
NMT-TY0566
[H]N([H])c1ccc(S(=O)(=O)N([H])c2cnc(N([H])[H])nc2N([H])[H])cc1
T07
native IFP available
T07
dockmulti_91311c650f2e_T07
0.884 1.000 0.668 native_similarity final_rank_score -29.8488 -1.62516 16 8 Pose
NMT-TY0566
[H]N([H])c1ccc(S(=O)(=O)N([H])c2cnc(N([H])[H])nc2N([H])[H])cc1
T03
native IFP available
T03
dockmulti_91311c650f2e_T03
0.843 1.000 0.550 native_similarity final_rank_score -27.3765 -1.51737 15 9 Pose
NMT-TY0566
[H]N([H])c1ccc(S(=O)(=O)N([H])c2cnc(N([H])[H])nc2N([H])[H])cc1
T15
native IFP available
T15
dockmulti_91311c650f2e_T15
0.804 1.000 0.441 native_similarity final_rank_score -20.2293 -1.19415 16 7 Pose
NMT-TY0566
[H]N([H])c1ccc(S(=O)(=O)N([H])c2cnc(N([H])[H])nc2N([H])[H])cc1
T16
native IFP available
T16
dockmulti_91311c650f2e_T16
0.758 1.000 0.308 native_similarity final_rank_score -21.4516 -1.26937 16 9 Pose