FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB Docking_panel_21Explorer results are being read from this database.
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2 compounds in matrix 5 best compound-target hits listed 5 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T02T06T08T12T14
MK152
[H]Oc1ccc(CCn2cc(COC[C@]3(C)CCc4c(C)c(O[H])c(C)c(C)c4O3)nn2)cc1O[H]
0.922 0.889 2 0.86 0.92
MK152
[H]Oc1ccc(CCn2cc(COC[C@@]3(C)CCc4c(C)c(O[H])c(C)c(C)c4O3)nn2)cc1O[H]
0.819 0.803 3 0.82 0.81 0.77

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
MK152
[H]Oc1ccc(CCn2cc(COC[C@]3(C)CCc4c(C)c(O[H])c(C)c(C)c4O3)nn2)cc1O[H]
T12
native IFP available
T12
dockmulti_91311c650f2e_T12
0.922 1.000 0.777 native_similarity final_rank_score -22.9301 -0.823637 18 11 Pose
MK152
[H]Oc1ccc(CCn2cc(COC[C@]3(C)CCc4c(C)c(O[H])c(C)c(C)c4O3)nn2)cc1O[H]
T08
native IFP available
T08
dockmulti_91311c650f2e_T08
0.857 1.000 0.591 native_similarity final_rank_score -25.285 -1.0212 20 5 Pose
MK152
[H]Oc1ccc(CCn2cc(COC[C@@]3(C)CCc4c(C)c(O[H])c(C)c(C)c4O3)nn2)cc1O[H]
T02
native IFP available
T02
dockmulti_91311c650f2e_T02
0.819 1.000 0.484 native_similarity final_rank_score -17.6699 -0.726869 18 3 Pose
MK152
[H]Oc1ccc(CCn2cc(COC[C@@]3(C)CCc4c(C)c(O[H])c(C)c(C)c4O3)nn2)cc1O[H]
T06
native IFP available
T06
dockmulti_91311c650f2e_T06
0.815 1.000 0.470 native_similarity final_rank_score -16.6012 -0.791369 20 4 Pose
MK152
[H]Oc1ccc(CCn2cc(COC[C@@]3(C)CCc4c(C)c(O[H])c(C)c(C)c4O3)nn2)cc1O[H]
T14
native IFP available
T14
dockmulti_91311c650f2e_T14
0.774 1.000 0.353 native_similarity final_rank_score -10.7425 -0.657314 17 9 Pose