FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB Docking_panel_21Explorer results are being read from this database.
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3 compounds in matrix 5 best compound-target hits listed 5 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T03T07T09T11T12
KB_chagas_219
[H]n1cc(C[N@@+]2([H])CCC[C@@H](c3cc(C(F)(F)F)n4ncnc4n3)C2)c2ccccc21
0.922 0.882 3 0.89 0.83 0.92
KB_chagas_219
[H]n1cc(CN2CCC[C@H](c3cc(C(F)(F)F)n4ncnc4n3)C2)c2ccccc21
0.875 0.875 1 0.87
KB_chagas_219
[H]n1cc(C[N@@+]2([H])CCC[C@H](c3cc(C(F)(F)F)n4ncnc4n3)C2)c2ccccc21
0.845 0.845 1 0.85

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
KB_chagas_219
[H]n1cc(C[N@@+]2([H])CCC[C@@H](c3cc(C(F)(F)F)n4ncnc4n3)C2)c2ccccc21
T12
native IFP available
T12
dockmulti_91311c650f2e_T12
0.922 1.000 0.777 native_similarity final_rank_score -27.5158 -0.968212 18 8 Pose
KB_chagas_219
[H]n1cc(C[N@@+]2([H])CCC[C@@H](c3cc(C(F)(F)F)n4ncnc4n3)C2)c2ccccc21
T03
native IFP available
T03
dockmulti_91311c650f2e_T03
0.895 1.000 0.699 native_similarity final_rank_score -23.4413 -0.895794 18 3 Pose
KB_chagas_219
[H]n1cc(CN2CCC[C@H](c3cc(C(F)(F)F)n4ncnc4n3)C2)c2ccccc21
T07
native IFP available
T07
dockmulti_91311c650f2e_T07
0.875 1.000 0.643 native_similarity final_rank_score -27.683 -0.971706 17 4 Pose
KB_chagas_219
[H]n1cc(C[N@@+]2([H])CCC[C@H](c3cc(C(F)(F)F)n4ncnc4n3)C2)c2ccccc21
T11
native IFP available
T11
dockmulti_91311c650f2e_T11
0.845 1.000 0.558 native_similarity final_rank_score -15.4041 -0.695357 11 4 Pose
KB_chagas_219
[H]n1cc(C[N@@+]2([H])CCC[C@@H](c3cc(C(F)(F)F)n4ncnc4n3)C2)c2ccccc21
T09
native IFP available
T09
dockmulti_91311c650f2e_T09
0.831 1.000 0.517 native_similarity final_rank_score -21.3478 -0.78349 14 1 Pose