FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB fairmolExplorer results are being read from this database.
Reset
2 compounds in matrix 3 best compound-target hits listed 3 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T08T16T19
KB_Leish_93
[H]O[C@H]1CCCN(c2cc(-c3ccccn3)nc(N([H])c3ccc(C)cc3)n2)C1
0.790 0.761 2 0.79 0.73
KB_Leish_93
[H]O[C@@H]1CCCN(c2cc(-c3ccccn3)nc(N([H])c3ccc(C)cc3)n2)C1
0.756 0.756 1 0.76

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
KB_Leish_93
[H]O[C@H]1CCCN(c2cc(-c3ccccn3)nc(N([H])c3ccc(C)cc3)n2)C1
T08
native IFP available
T08
selection_import_t08
0.790 1.000 0.399 native_similarity final_rank_score -27.6681 -1.18942 10 8 Pose
KB_Leish_93
[H]O[C@@H]1CCCN(c2cc(-c3ccccn3)nc(N([H])c3ccc(C)cc3)n2)C1
T16
native IFP available
T16
selection_import_t16
0.756 1.000 0.302 native_similarity final_rank_score -18.0943 -0.896782 17 5 Pose
KB_Leish_93
[H]O[C@H]1CCCN(c2cc(-c3ccccn3)nc(N([H])c3ccc(C)cc3)n2)C1
T19
native IFP available
T19
selection_import_t19
0.732 1.000 0.234 native_similarity final_rank_score -34.5559 -1.3108 21 9 Pose