FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB Docking_panel_21Explorer results are being read from this database.
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2 compounds in matrix 6 best compound-target hits listed 6 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T08T12T14T15T18T20
KB_Leish_74
[H]O[C@H]1CN(CCc2c(Cl)cnc3ccc(OC)nc23)CC[C@@H]1[N+]([H])([H])Cc1cc2c(cn1)OCS2
0.891 0.875 2 0.89 0.86
KB_Leish_74
[H]O[C@H]1C[N@+]([H])(CCc2c(Cl)cnc3ccc(OC)nc23)CC[C@@H]1[N+]([H])([H])Cc1cc2c(cn1)OCS2
0.877 0.815 4 0.88 0.80 0.82 0.76

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
KB_Leish_74
[H]O[C@H]1CN(CCc2c(Cl)cnc3ccc(OC)nc23)CC[C@@H]1[N+]([H])([H])Cc1cc2c(cn1)OCS2
T08
native IFP available
T08
dockmulti_91311c650f2e_T08
0.891 1.000 0.690 native_similarity final_rank_score -29.3973 -1.04599 18 6 Pose
KB_Leish_74
[H]O[C@H]1C[N@+]([H])(CCc2c(Cl)cnc3ccc(OC)nc23)CC[C@@H]1[N+]([H])([H])Cc1cc2c(cn1)OCS2
T12
native IFP available
T12
dockmulti_91311c650f2e_T12
0.877 1.000 0.647 native_similarity final_rank_score -20.8378 -0.74759 16 8 Pose
KB_Leish_74
[H]O[C@H]1CN(CCc2c(Cl)cnc3ccc(OC)nc23)CC[C@@H]1[N+]([H])([H])Cc1cc2c(cn1)OCS2
T15
native IFP available
T15
dockmulti_91311c650f2e_T15
0.859 1.000 0.597 native_similarity final_rank_score -21.9316 -0.77501 14 5 Pose
KB_Leish_74
[H]O[C@H]1C[N@+]([H])(CCc2c(Cl)cnc3ccc(OC)nc23)CC[C@@H]1[N+]([H])([H])Cc1cc2c(cn1)OCS2
T18
native IFP available
T18
dockmulti_91311c650f2e_T18
0.820 1.000 0.485 native_similarity final_rank_score -21.4915 -0.544373 9 3 Pose
KB_Leish_74
[H]O[C@H]1C[N@+]([H])(CCc2c(Cl)cnc3ccc(OC)nc23)CC[C@@H]1[N+]([H])([H])Cc1cc2c(cn1)OCS2
T14
native IFP available
T14
dockmulti_91311c650f2e_T14
0.802 1.000 0.434 native_similarity final_rank_score -14.6839 -0.656243 18 5 Pose
KB_Leish_74
[H]O[C@H]1C[N@+]([H])(CCc2c(Cl)cnc3ccc(OC)nc23)CC[C@@H]1[N+]([H])([H])Cc1cc2c(cn1)OCS2
T20
native IFP available
T20
dockmulti_91311c650f2e_T20
0.762 1.000 0.321 native_similarity final_rank_score -15.9399 -0.53287 12 5 Pose