FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB Docking_panel_21Explorer results are being read from this database.
Reset
2 compounds in matrix 4 best compound-target hits listed 4 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T02T11T19T20
KB_Leish_101
[H]N(c1ccc(C)cn1)c1nc([C@H]2CCC[N@+]2([H])Cc2ccn([H])n2)cs1
0.898 0.891 3 0.89 0.89 0.90
KB_Leish_101
[H]N(c1ccc(C)cn1)c1nc([C@@H]2CCC[N@@+]2([H])Cc2ccn([H])n2)cs1
0.733 0.733 1 0.73

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
KB_Leish_101
[H]N(c1ccc(C)cn1)c1nc([C@H]2CCC[N@+]2([H])Cc2ccn([H])n2)cs1
T20
native IFP available
T20
dockmulti_91311c650f2e_T20
0.898 1.000 0.710 native_similarity final_rank_score -16.5271 -0.627171 11 5 Pose
KB_Leish_101
[H]N(c1ccc(C)cn1)c1nc([C@H]2CCC[N@+]2([H])Cc2ccn([H])n2)cs1
T02
native IFP available
T02
dockmulti_91311c650f2e_T02
0.887 1.000 0.677 native_similarity final_rank_score -23.8342 -0.883699 20 2 Pose
KB_Leish_101
[H]N(c1ccc(C)cn1)c1nc([C@H]2CCC[N@+]2([H])Cc2ccn([H])n2)cs1
T11
native IFP available
T11
dockmulti_91311c650f2e_T11
0.886 1.000 0.676 native_similarity final_rank_score -27.4014 -1.05673 13 8 Pose
KB_Leish_101
[H]N(c1ccc(C)cn1)c1nc([C@@H]2CCC[N@@+]2([H])Cc2ccn([H])n2)cs1
T19
native IFP available
T19
dockmulti_91311c650f2e_T19
0.733 1.000 0.238 native_similarity final_rank_score -33.262 -1.21782 19 5 Pose