FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB Docking_panel_21Explorer results are being read from this database.
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2 compounds in matrix 4 best compound-target hits listed 4 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T02T03T09T16
KB_HAT_148
[H][N+]1(Cc2ccc(NS(=O)(=O)c3ccc(C)cc3)cc2)CCN(C(=O)c2cccc(C)c2)CC1
0.860 0.826 3 0.86 0.83 0.79
KB_HAT_148
[H]N(c1ccc(CN2CCN(C(=O)c3cccc(C)c3)CC2)cc1)S(=O)(=O)c1ccc(C)cc1
0.804 0.804 1 0.80

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
KB_HAT_148
[H][N+]1(Cc2ccc(NS(=O)(=O)c3ccc(C)cc3)cc2)CCN(C(=O)c2cccc(C)c2)CC1
T02
native IFP available
T02
dockmulti_91311c650f2e_T02
0.860 1.000 0.600 native_similarity final_rank_score -19.878 -0.713616 18 2 Pose
KB_HAT_148
[H][N+]1(Cc2ccc(NS(=O)(=O)c3ccc(C)cc3)cc2)CCN(C(=O)c2cccc(C)c2)CC1
T03
native IFP available
T03
dockmulti_91311c650f2e_T03
0.830 1.000 0.513 native_similarity final_rank_score -26.1485 -0.762494 17 3 Pose
KB_HAT_148
[H]N(c1ccc(CN2CCN(C(=O)c3cccc(C)c3)CC2)cc1)S(=O)(=O)c1ccc(C)cc1
T16
native IFP available
T16
dockmulti_91311c650f2e_T16
0.804 1.000 0.440 native_similarity final_rank_score -23.9087 -0.782252 19 2 Pose
KB_HAT_148
[H][N+]1(Cc2ccc(NS(=O)(=O)c3ccc(C)cc3)cc2)CCN(C(=O)c2cccc(C)c2)CC1
T09
native IFP available
T09
dockmulti_91311c650f2e_T09
0.788 1.000 0.394 native_similarity final_rank_score -23.5859 -0.829986 17 2 Pose