FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB Docking_panel_21Explorer results are being read from this database.
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3 compounds in matrix 4 best compound-target hits listed 4 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T08T16T19T20
KB_HAT_101
[H]N([H])C(=O)[C@@H]1CCN1c1nc(CCCC)cc(N([H])c2cc(C3CCC3)n([H])n2)n1
0.945 0.945 1 0.94
KB_HAT_101
[H]N([H])C(=O)[C@H]1CCN1c1nc(CCCC)cc(N([H])c2cc(C3CCC3)n([H])n2)[n+]1[H]
0.858 0.819 2 0.86 0.78
KB_HAT_101
[H]N([H])C(=O)[C@@H]1CCN1c1nc(CCCC)cc(N([H])c2cc(C3CCC3)n([H])n2)[n+]1[H]
0.739 0.739 1 0.74

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
KB_HAT_101
[H]N([H])C(=O)[C@@H]1CCN1c1nc(CCCC)cc(N([H])c2cc(C3CCC3)n([H])n2)n1
T20
native IFP available
T20
dockmulti_91311c650f2e_T20
0.945 1.000 0.842 native_similarity final_rank_score -13.198 -0.59348 9 4 Pose
KB_HAT_101
[H]N([H])C(=O)[C@H]1CCN1c1nc(CCCC)cc(N([H])c2cc(C3CCC3)n([H])n2)[n+]1[H]
T08
native IFP available
T08
dockmulti_91311c650f2e_T08
0.858 1.000 0.596 native_similarity final_rank_score -24.6899 -1.1599 17 6 Pose
KB_HAT_101
[H]N([H])C(=O)[C@H]1CCN1c1nc(CCCC)cc(N([H])c2cc(C3CCC3)n([H])n2)[n+]1[H]
T16
native IFP available
T16
dockmulti_91311c650f2e_T16
0.779 1.000 0.368 native_similarity final_rank_score -14.8629 -0.833103 15 6 Pose
KB_HAT_101
[H]N([H])C(=O)[C@@H]1CCN1c1nc(CCCC)cc(N([H])c2cc(C3CCC3)n([H])n2)[n+]1[H]
T19
native IFP available
T19
dockmulti_91311c650f2e_T19
0.739 1.000 0.255 native_similarity final_rank_score -29.8721 -1.16167 19 9 Pose