FAIRMol

Reverse docking explorer

Search one compound across many targets or scan the strongest compound-target pairs in the active database. The combined reverse-docking score uses a normalized docking-score estimator together with an interaction-fingerprint component.

DB Docking_panel_21Explorer results are being read from this database.
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5 compounds in matrix 9 best compound-target hits listed 6 targets
• Combined reverse-docking score = 65% normalized docking-score estimator + 35% interaction-fingerprint component.
• When a native ligand exists for an experiment, the interaction-fingerprint component is driven by similarity to the native contact/H-bond pattern.
• When no native ligand exists, the interaction-fingerprint component falls back to contact richness within the experiment (normalized contacts and H-bonds).

Compounds × targets matrix

Each cell shows the best combined reverse-docking score found for that compound on that target. Blank cells mean no imported pose passed the current filters.
Compound Best Mean Targets T08T09T11T15T19T21
GemmaOHDUnisi_3
[H]OB(O[H])c1ccc(C(=O)N([H])c2ccc(OC)c(S(=O)(=O)N([H])c3ccc(OC)cc3)c2)s1
0.893 0.893 1 0.89
GemmaOHDUnisi_36
[H]Oc1ccc(-c2cc3cc(/C=C/C(=O)c4ccc(O[H])cc4O[H])ccc3n2C)cc1
0.886 0.795 3 0.80 0.70 0.89
GemmaOHDUnisi_38
[H]Oc1ccc(C(=O)/C=C/c2ccc3oc(-c4ccccc4)cc3c2)c(O)c1
0.880 0.823 3 0.80 0.79 0.88
GemmaOHDUnisi_30
[H]Oc1ccc(C(=O)/C=C/c2ccc3c(ccn3[H])c2)c(O)c1
0.784 0.784 1 0.78
GemmaOHDUnisi_34
[H]Oc1ccc(-c2cc3cc(/C=C/C(=O)c4ccccc4)ccc3o2)cc1
0.751 0.751 1 0.75

Best compound-target hits

The score column is the combined reverse-docking score. The next two columns expose its components: normalized score-estimator and interaction fingerprint.
CompoundTargetExperimentCombinedScore partIFP partIFP modeMetricDock scoreInter normContactsHB
GemmaOHDUnisi_3
[H]OB(O[H])c1ccc(C(=O)N([H])c2ccc(OC)c(S(=O)(=O)N([H])c3ccc(OC)cc3)c2)s1
T11
native IFP available
T11
dockmulti_91311c650f2e_T11
0.893 1.000 0.695 native_similarity final_rank_score -18.4651 -0.781534 17 5 Pose
GemmaOHDUnisi_36
[H]Oc1ccc(-c2cc3cc(/C=C/C(=O)c4ccc(O[H])cc4O[H])ccc3n2C)cc1
T21
native IFP available
T21
dockmulti_91311c650f2e_T21
0.886 1.000 0.674 native_similarity final_rank_score -22.6513 -0.81077 14 7 Pose
GemmaOHDUnisi_38
[H]Oc1ccc(C(=O)/C=C/c2ccc3oc(-c4ccccc4)cc3c2)c(O)c1
T21
native IFP available
T21
dockmulti_91311c650f2e_T21
0.880 1.000 0.656 native_similarity final_rank_score -20.5123 -0.68663 15 5 Pose
GemmaOHDUnisi_36
[H]Oc1ccc(-c2cc3cc(/C=C/C(=O)c4ccc(O[H])cc4O[H])ccc3n2C)cc1
T08
native IFP available
T08
dockmulti_91311c650f2e_T08
0.799 1.000 0.425 native_similarity final_rank_score -26.92 -1.02158 15 4 Pose
GemmaOHDUnisi_38
[H]Oc1ccc(C(=O)/C=C/c2ccc3oc(-c4ccccc4)cc3c2)c(O)c1
T08
native IFP available
T08
dockmulti_91311c650f2e_T08
0.797 1.000 0.419 native_similarity final_rank_score -32.3744 -1.26118 13 6 Pose
GemmaOHDUnisi_38
[H]Oc1ccc(C(=O)/C=C/c2ccc3oc(-c4ccccc4)cc3c2)c(O)c1
T11
native IFP available
T11
dockmulti_91311c650f2e_T11
0.793 1.000 0.409 native_similarity final_rank_score -23.6271 -0.956451 17 4 Pose
GemmaOHDUnisi_30
[H]Oc1ccc(C(=O)/C=C/c2ccc3c(ccn3[H])c2)c(O)c1
T09
native IFP available
T09
dockmulti_91311c650f2e_T09
0.784 1.000 0.383 native_similarity final_rank_score -24.1471 -1.17601 15 5 Pose
GemmaOHDUnisi_34
[H]Oc1ccc(-c2cc3cc(/C=C/C(=O)c4ccccc4)ccc3o2)cc1
T15
native IFP available
T15
dockmulti_91311c650f2e_T15
0.751 1.000 0.289 native_similarity final_rank_score -23.0506 -0.903914 16 1 Pose
GemmaOHDUnisi_36
[H]Oc1ccc(-c2cc3cc(/C=C/C(=O)c4ccc(O[H])cc4O[H])ccc3n2C)cc1
T19
native IFP available
T19
dockmulti_91311c650f2e_T19
0.702 1.000 0.148 native_similarity final_rank_score -28.1075 -0.949378 20 5 Pose