FAIRMol

Z16027953

Pose ID 9741 Compound 1203 Pose 1162

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Good LE (-0.315 kcal/mol/HA) ✓ Good fit quality (FQ -3.01) ✓ Good H-bonds (4 bonds) ✗ Very high strain energy (26.0 kcal/mol) ✗ Geometry warnings ✗ Protein contact clashes ℹ SASA not computed
Score
-9.133
kcal/mol
LE
-0.315
kcal/mol/HA
Fit Quality
-3.01
FQ (Leeson)
HAC
29
heavy atoms
MW
394
Da
LogP
2.53
cLogP
Strain ΔE
26.0 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: good
Geometry reliability: low
Reason: geometry warning, clashes, protein contact clashes, strain 26.0 kcal/mol

Interaction summary

Collapsible panels
H-bonds 4 Hydrophobic 24 π–π 3 Clashes 10 Severe clashes 0
Final rank6.444413830024239Score-9.13326
Inter norm-0.835369Intra norm0.497599
Top1000noExcludedno
Contacts17H-bonds4
Artifact reasongeometry warning; 11 clashes; 10 protein contact clashes; high strain Δ 42.3
ResiduesA:ALA34;A:ARG59;A:ASP54;A:GLN56;A:GLY161;A:ILE160;A:ILE47;A:LEU90;A:LEU97;A:MET55;A:NDP301;A:PHE58;A:PHE94;A:PRO91;A:TYR166;A:VAL32;A:VAL33

Protein summary

223 residues
Protein targetT06Atoms3452
Residues223Chains1
Residue summaryARG:408; VAL:352; LYS:308; LEU:304; PRO:238; ILE:209; GLU:195; THR:182; SER:176; ALA:160; PHE:140; ASN:126; GLY:126; ASP:108; GLN:85; NDP:74

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name8RHTContacts21
PoseOpen native poseH-bonds6
IFP residuesA:ALA34; A:ASP54; A:HIS182; A:ILE160; A:ILE47; A:LEU90; A:LEU97; A:MET55; A:NDP301; A:PHE233; A:PHE58; A:PHE94; A:PRO91; A:SER89; A:THR184; A:THR86; A:TRP49; A:TYR166; A:TYR57; A:VAL32; A:VAL33
Current overlap14Native recall0.67
Jaccard0.58RMSD-
H-bond strict0Strict recall0.00
H-bond same residue+role0Role recall0.00
H-bond same residue0Residue recall0.00

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
1077 5.003438419027329 -1.04612 -27.0807 11 23 0 0.00 0.00 - no Open
1604 5.1910895123134075 -0.815377 -21.9974 6 15 1 0.05 0.00 - no Open
1608 5.33148680171199 -0.767169 -27.1261 7 16 1 0.05 0.00 - no Open
1163 5.551448951917198 -0.77159 -16.3561 4 16 14 0.67 0.00 - no Open
1605 5.595679038556167 -0.763376 -19.0878 5 21 1 0.05 0.00 - no Open
1698 5.762804483422982 -0.580681 -8.8695 9 14 0 0.00 0.00 - no Open
1606 5.931587814186224 -0.628975 -14.4266 6 18 1 0.05 0.00 - no Open
1164 6.094346852211321 -0.766971 -10.1997 3 18 16 0.76 0.00 - no Open
1162 6.444413830024239 -0.835369 -9.13326 4 17 14 0.67 0.00 - no Current
1166 6.475041900743294 -0.836178 -14.6246 4 16 14 0.67 0.00 - no Open
1695 6.640473401922036 -0.750944 -17.3946 7 12 0 0.00 0.00 - no Open
1194 7.497948552462457 -0.989691 -18.8202 7 14 0 0.00 0.00 - no Open
1607 6.386067244284125 -0.781274 -20.0784 3 17 1 0.05 0.00 - yes Open
1693 6.862943417541378 -0.607459 -13.793 8 17 0 0.00 0.00 - yes Open
1081 7.351840382609471 -0.99993 -24.2698 9 23 0 0.00 0.00 - yes Open
1193 8.30331011879626 -1.03911 -20.7889 8 20 0 0.00 0.00 - yes Open
1694 8.838393030440574 -0.646642 -17.0159 6 16 0 0.00 0.00 - yes Open
1198 8.936511162310344 -0.9705 -20.3664 8 15 0 0.00 0.00 - yes Open
1603 9.05979073358385 -0.745663 -19.6442 12 16 1 0.05 0.00 - yes Open
1195 9.180771122448231 -0.98797 -20.7422 7 20 0 0.00 0.00 - yes Open
1197 9.58358171648457 -0.901259 -8.96109 9 17 0 0.00 0.00 - yes Open
1076 9.681030475258796 -0.933328 -19.2815 6 19 0 0.00 0.00 - yes Open
1697 9.696589521284785 -0.583552 -16.0209 7 14 0 0.00 0.00 - yes Open
1696 10.07190966349914 -0.726935 -18.2131 9 16 0 0.00 0.00 - yes Open
1196 10.208847296040425 -0.977842 -16.8413 4 13 0 0.00 0.00 - yes Open
1080 10.389098008978085 -1.07129 -19.5439 6 19 0 0.00 0.00 - yes Open
1078 11.897146124212874 -1.01195 -18.6481 8 19 0 0.00 0.00 - yes Open
1079 12.37917067131761 -0.953674 -14.2889 8 19 0 0.00 0.00 - yes Open
1165 12.644067386113937 -0.776387 -2.86358 4 15 13 0.62 0.00 - yes Open
1167 12.696086250357059 -0.73911 -10.8795 5 17 15 0.71 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -9.133kcal/mol
Ligand efficiency (LE) -0.3149kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -3.006
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 29HA

Physicochemical properties

Molecular weight 394.4Da
Lipinski: ≤ 500 Da
LogP (cLogP) 2.53
Lipinski: ≤ 5
Rotatable bonds 5

Conformational strain (MMFF94s)

Strain energy (ΔE) 26.01kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 85.51kcal/mol
Minimised FF energy 59.50kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.