FAIRMol

OSA_Lib_43

Pose ID 918 Compound 333 Pose 918

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Excellent LE (-0.716 kcal/mol/HA) ✓ Good fit quality (FQ -7.27) ✓ Good H-bonds (3 bonds) ✗ Very high strain energy (39.1 kcal/mol) ✗ Geometry warnings ℹ SASA not computed
Score
-25.765
kcal/mol
LE
-0.716
kcal/mol/HA
Fit Quality
-7.27
FQ (Leeson)
HAC
36
heavy atoms
MW
491
Da
LogP
1.74
cLogP
Strain ΔE
39.1 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, strain 39.1 kcal/mol

Interaction summary

Collapsible panels
H-bonds 3 Hydrophobic 24 π–π 2 Clashes 16 Severe clashes 2
Final rank60.39014575474776Score-25.7652
Inter norm-0.715514Intra norm-0.000187178
Top1000noExcludedyes
Contacts21H-bonds3
Artifact reasonexcluded; geometry warning; 18 clashes; 2 protein clashes
ResiduesA:ALA10;A:ASN65;A:ASP22;A:GLU31;A:GLY21;A:ILE61;A:ILE8;A:LEU23;A:LEU28;A:LEU68;A:NAP201;A:PHE32;A:PHE35;A:PRO27;A:PRO62;A:SER60;A:THR57;A:TRP25;A:TYR122;A:VAL116;A:VAL9

Protein summary

200 residues
Protein targetT02Atoms3128
Residues200Chains2
Residue summaryLYS:374; LEU:361; GLU:240; VAL:224; ARG:192; PHE:180; ILE:171; PRO:168; ASN:140; SER:132; TYR:126; GLN:119; ASP:108; MET:102; THR:98; GLY:91

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name5SD8Contacts21
PoseOpen native poseH-bonds5
IFP residuesA:ALA10; A:ASN65; A:ASP22; A:GLN36; A:GLU31; A:GLY117; A:GLY21; A:ILE61; A:ILE8; A:LEU23; A:LEU68; A:NAP201; A:PHE32; A:PHE35; A:PRO62; A:SER60; A:THR137; A:THR57; A:TYR122; A:VAL116; A:VAL9
Current overlap18Native recall0.86
Jaccard0.75RMSD-
H-bond strict0Strict recall0.00
H-bond same residue+role0Role recall0.00
H-bond same residue0Residue recall0.00

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
960 4.826503894865375 -0.656051 -22.8818 3 17 0 0.00 0.00 - no Open
919 5.808082337017025 -0.575939 -17.5908 3 15 10 0.48 0.20 - no Open
958 5.9117766679857615 -0.534388 -16.3143 4 14 0 0.00 0.00 - no Open
975 6.21047578831829 -0.457542 -10.9767 3 14 0 0.00 0.00 - no Open
976 6.245710768749463 -0.538356 -19.0736 4 11 0 0.00 0.00 - no Open
921 6.564751731567194 -0.614055 -22.2168 4 17 14 0.67 0.40 - no Open
966 6.588736720845645 -0.56841 -17.7307 5 14 0 0.00 0.00 - no Open
927 7.923351763023396 -0.559531 -18.2833 2 20 18 0.86 0.00 - no Open
959 55.16845693170977 -0.599004 -18.9095 3 16 0 0.00 0.00 - no Open
965 55.39037580418941 -0.519079 -18.0533 3 13 0 0.00 0.00 - no Open
964 55.4547426689101 -0.549954 -19.4114 2 12 0 0.00 0.00 - no Open
971 56.4560103950494 -0.516542 -11.9404 5 13 0 0.00 0.00 - no Open
930 56.94094499893816 -0.72047 -7.77951 1 21 19 0.90 0.00 - no Open
978 9.398886030570841 -0.561908 -7.24905 3 17 0 0.00 0.00 - yes Open
924 56.250375098920614 -0.532772 -8.05381 0 18 17 0.81 0.00 - yes Open
969 56.26096785719301 -0.631283 -21.1711 2 16 0 0.00 0.00 - yes Open
970 56.27280601729279 -0.574895 -16.4472 2 14 0 0.00 0.00 - yes Open
920 56.39425801769821 -0.569045 -16.4935 0 19 16 0.76 0.00 - yes Open
925 56.464474361735 -0.541189 -14.8007 2 18 13 0.62 0.00 - yes Open
931 56.564016733625934 -0.511389 -15.7556 1 12 8 0.38 0.00 - yes Open
963 56.83044584149283 -0.473946 -15.8629 1 17 0 0.00 0.00 - yes Open
961 57.383183121750804 -0.642125 -22.6918 2 16 0 0.00 0.00 - yes Open
972 57.39817307960844 -0.467829 -16.2853 1 17 0 0.00 0.00 - yes Open
967 57.52984142300179 -0.625508 -18.8171 3 17 0 0.00 0.00 - yes Open
973 57.626119157043455 -0.621989 -22.8404 2 17 0 0.00 0.00 - yes Open
962 57.675130763308104 -0.640697 -22.7533 3 15 0 0.00 0.00 - yes Open
968 57.724646291174565 -0.622439 -22.022 4 17 0 0.00 0.00 - yes Open
923 57.74052012191032 -0.699627 -17.1276 2 20 16 0.76 0.00 - yes Open
974 57.97259049224995 -0.605685 -20.6048 2 17 0 0.00 0.00 - yes Open
977 58.131462184730054 -0.697339 -22.1539 4 15 0 0.00 0.00 - yes Open
929 58.25766722607442 -0.587102 -15.5101 1 20 17 0.81 0.20 - yes Open
981 58.72917371361217 -0.423748 -14.1372 2 12 0 0.00 0.00 - yes Open
917 58.74059449031091 -0.634513 -22.3278 3 18 14 0.67 0.20 - yes Open
979 58.93046332164697 -0.648465 -18.8427 6 16 0 0.00 0.00 - yes Open
928 59.40816438757014 -0.58568 -12.5864 5 21 17 0.81 0.40 - yes Open
980 59.532216229383934 -0.516104 -19.7186 3 17 0 0.00 0.00 - yes Open
922 59.8284064671385 -0.613179 -15.3558 4 24 20 0.95 0.20 - yes Open
932 60.089461716634666 -0.621729 -12.0536 1 17 17 0.81 0.20 - yes Open
918 60.39014575474776 -0.715514 -25.7652 3 21 18 0.86 0.00 - yes Current
926 62.67347159229395 -0.675274 -10.1422 2 21 18 0.86 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -25.765kcal/mol
Ligand efficiency (LE) -0.7157kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -7.274
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 36HA

Physicochemical properties

Molecular weight 490.7Da
Lipinski: ≤ 500 Da
LogP (cLogP) 1.74
Lipinski: ≤ 5
Rotatable bonds 6

Conformational strain (MMFF94s)

Strain energy (ΔE) 39.13kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 127.00kcal/mol
Minimised FF energy 87.87kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.