FAIRMol

Z266766868

Pose ID 7670 Compound 862 Pose 1083

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Good H-bonds (4 bonds) ✗ Very high strain energy (25.8 kcal/mol) ✗ Poor LE (-0.100 kcal/mol/HA) ✗ Geometry warnings ℹ SASA not computed
Score
-2.391
kcal/mol
LE
-0.100
kcal/mol/HA
Fit Quality
-0.89
FQ (Leeson)
HAC
24
heavy atoms
MW
343
Da
LogP
3.53
cLogP
Strain ΔE
25.8 kcal/mol
SASA buried
computing…
Overall: Likely artefact or unreliable pose
Binding evidence: weak
Native-like contacts: strong
Ligand efficiency: weak
Geometry reliability: low
Reason: geometry warning, clashes, strain 25.8 kcal/mol

Interaction summary

Collapsible panels
H-bonds 4 Hydrophobic 14 π–π 2 Clashes 20 Severe clashes 1
Final rank10.295575461154481Score-2.3908
Inter norm-0.730822Intra norm0.631205
Top1000noExcludedyes
Contacts12H-bonds4
Artifact reasonexcluded; hard geometry fail; 1 severe clash; 1 protein clash; high normalized intra; high strain Δ 30.6
ResiduesA:ARG17;A:GLY225;A:HIS241;A:LEU188;A:LEU226;A:LEU229;A:NDP302;A:PHE113;A:SER111;A:TYR194;A:TYR283;D:ARG287

Protein summary

308 residues
Protein targetT04Atoms4210
Residues308Chains3
Residue summaryLEU:494; ALA:421; ARG:384; VAL:368; THR:295; TYR:231; SER:198; PRO:196; ILE:190; LYS:176; ASN:154; GLU:150; GLY:126; PHE:120; HIS:119; ASP:108

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name7PXXContacts19
PoseOpen native poseH-bonds8
IFP residuesA:ARG17; A:ASP181; A:GLY225; A:HIS241; A:LEU188; A:LEU226; A:LEU229; A:LYS198; A:MET233; A:NDP302; A:PHE113; A:PRO115; A:SER111; A:SER112; A:SER227; A:TYR191; A:TYR194; A:VAL230; D:ARG287
Current overlap11Native recall0.58
Jaccard0.55RMSD-
H-bond strict0Strict recall0.00
H-bond same residue+role0Role recall0.00
H-bond same residue0Residue recall0.00

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
1085 3.359753612037696 -0.744035 -33.7684 0 12 11 0.58 0.00 - no Open
1084 3.6964274695136785 -1.01986 -41.1289 0 14 13 0.68 0.00 - no Open
1089 4.0110527975039005 -0.698038 -11.6276 0 13 12 0.63 0.00 - no Open
1081 6.877864207759705 -0.702507 -7.65221 2 12 12 0.63 0.00 - no Open
1086 4.54715210133792 -0.936536 -18.442 3 13 13 0.68 0.00 - yes Open
1082 4.5504073924947335 -1.04565 -21.6751 2 12 12 0.63 0.00 - yes Open
1088 4.72320468939807 -0.948376 -19.6837 3 12 12 0.63 0.00 - yes Open
1080 4.83042990372482 -0.946502 -17.5927 3 11 11 0.58 0.00 - yes Open
1087 5.8246081240266685 -0.654434 -12.4506 0 11 11 0.58 0.00 - yes Open
1083 10.295575461154481 -0.730822 -2.3908 4 12 11 0.58 0.00 - yes Current

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -2.391kcal/mol
Ligand efficiency (LE) -0.0996kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -0.893
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 24HA

Physicochemical properties

Molecular weight 342.8Da
Lipinski: ≤ 500 Da
LogP (cLogP) 3.53
Lipinski: ≤ 5
Rotatable bonds 5

Conformational strain (MMFF94s)

Strain energy (ΔE) 25.79kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 82.86kcal/mol
Minimised FF energy 57.07kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.