FAIRMol

KB_Leish_101

Pose ID 720 Compound 7 Pose 720

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Weak Marginal quality. Consider only alongside better-scoring alternatives.
✓ Excellent LE (-1.064 kcal/mol/HA) ✓ Good fit quality (FQ -9.54) ✓ Good H-bonds (3 bonds) ✗ Very high strain energy (21.4 kcal/mol) ✗ Geometry warnings ℹ SASA not computed
Score
-25.538
kcal/mol
LE
-1.064
kcal/mol/HA
Fit Quality
-9.54
FQ (Leeson)
HAC
24
heavy atoms
MW
341
Da
LogP
2.23
cLogP
Strain ΔE
21.4 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, strain 21.4 kcal/mol

Interaction summary

Collapsible panels
H-bonds 3 Hydrophobic 22 π–π 1 Clashes 3 Severe clashes 1
Final rank52.612234295974275Score-25.538
Inter norm-0.891941Intra norm-0.17214
Top1000noExcludedyes
Contacts18H-bonds3
Artifact reasonexcluded; geometry warning; 4 clashes; 1 protein clash
ResiduesA:ALA10;A:ASP22;A:GLU31;A:GLY21;A:ILE61;A:ILE8;A:LEU23;A:LEU68;A:NAP201;A:PHE32;A:PHE35;A:PRO62;A:SER60;A:THR137;A:THR57;A:TYR122;A:VAL116;A:VAL9

Protein summary

200 residues
Protein targetT02Atoms3128
Residues200Chains2
Residue summaryLYS:374; LEU:361; GLU:240; VAL:224; ARG:192; PHE:180; ILE:171; PRO:168; ASN:140; SER:132; TYR:126; GLN:119; ASP:108; MET:102; THR:98; GLY:91

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name5SD8Contacts21
PoseOpen native poseH-bonds5
IFP residuesA:ALA10; A:ASN65; A:ASP22; A:GLN36; A:GLU31; A:GLY117; A:GLY21; A:ILE61; A:ILE8; A:LEU23; A:LEU68; A:NAP201; A:PHE32; A:PHE35; A:PRO62; A:SER60; A:THR137; A:THR57; A:TYR122; A:VAL116; A:VAL9
Current overlap18Native recall0.86
Jaccard0.86RMSD-
H-bond strict1Strict recall0.20
H-bond same residue+role1Role recall0.20
H-bond same residue1Residue recall0.20

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
717 2.206333458912313 -0.883699 -23.8342 2 20 19 0.90 0.20 - no Open
719 2.811728024846724 -1.02463 -29.1846 2 17 17 0.81 0.40 - no Open
508 2.9713068037673374 -1.05673 -27.4014 8 13 0 0.00 0.00 - no Open
718 3.349190829421271 -0.937615 -28.0142 2 18 18 0.86 0.20 - no Open
689 4.616306717670226 -0.627171 -16.5271 5 11 0 0.00 0.00 - no Open
506 3.723413214037131 -0.821855 -24.6354 3 17 0 0.00 0.00 - yes Open
504 4.373848278576643 -0.978027 -26.1159 8 14 0 0.00 0.00 - yes Open
690 4.5895314355052665 -0.65509 -18.5286 6 12 0 0.00 0.00 - yes Open
509 4.877034484710657 -0.99498 -26.4576 8 14 0 0.00 0.00 - yes Open
687 5.000415142517421 -0.843529 -22.6019 5 7 0 0.00 0.00 - yes Open
505 5.2088665555536355 -0.912245 -26.7049 2 17 0 0.00 0.00 - yes Open
510 6.217204623503973 -0.888423 -25.0004 8 14 0 0.00 0.00 - yes Open
720 52.612234295974275 -0.891941 -25.538 3 18 18 0.86 0.20 - yes Current
688 54.426005414082425 -0.738238 -22.1628 6 8 0 0.00 0.00 - yes Open
511 55.81278002637568 -0.977846 -25.4141 6 18 0 0.00 0.00 - yes Open
507 57.55189034350466 -0.935779 -24.1095 4 15 0 0.00 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -25.538kcal/mol
Ligand efficiency (LE) -1.0641kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -9.536
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 24HA

Physicochemical properties

Molecular weight 341.5Da
Lipinski: ≤ 500 Da
LogP (cLogP) 2.23
Lipinski: ≤ 5
Rotatable bonds 5

Conformational strain (MMFF94s)

Strain energy (ΔE) 21.44kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 30.11kcal/mol
Minimised FF energy 8.67kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.