FAIRMol

Z2786555116

Pose ID 6446 Compound 358 Pose 3128

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Excellent LE (-0.759 kcal/mol/HA) ✓ Good fit quality (FQ -7.33) ✓ Good H-bonds (4 bonds) ✗ Very high strain energy (26.1 kcal/mol) ✗ Geometry warnings ℹ SASA not computed
Score
-22.782
kcal/mol
LE
-0.759
kcal/mol/HA
Fit Quality
-7.33
FQ (Leeson)
HAC
30
heavy atoms
MW
421
Da
LogP
3.94
cLogP
Strain ΔE
26.1 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: mixed
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, strain 26.1 kcal/mol

Interaction summary

Collapsible panels
H-bonds 4 Hydrophobic 21 π–π 2 Clashes 13 Severe clashes 3
Final rank10.682020037457598Score-22.7817
Inter norm-0.875906Intra norm0.116516
Top1000noExcludedyes
Contacts13H-bonds4
Artifact reasonexcluded; geometry warning; 15 clashes; 3 protein clashes; high strain Δ 27.8
ResiduesA:ARG97;A:ILE45;A:LEU94;A:LYS57;A:LYS95;A:MET53;A:PHE56;A:PHE91;A:PRO50;A:PRO88;A:PRO93;A:THR54;A:VAL87

Protein summary

225 residues
Protein targetT03Atoms3428
Residues225Chains2
Residue summaryLEU:380; ARG:360; VAL:272; LYS:264; ALA:240; GLU:240; PRO:224; PHE:180; THR:154; ILE:152; SER:132; TYR:126; GLN:119; ASN:98; GLY:84; NDP:74

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name3CL9Contacts20
PoseOpen native poseH-bonds9
IFP residuesA:ALA32; A:ARG97; A:ASP52; A:ILE45; A:LEU94; A:LYS57; A:MET53; A:NDP301; A:PHE56; A:PHE91; A:PRO88; A:SER86; A:THR180; A:THR54; A:THR83; A:TYR162; A:VAL156; A:VAL30; A:VAL31; A:VAL87
Current overlap10Native recall0.50
Jaccard0.43RMSD-
H-bond strict2Strict recall0.29
H-bond same residue+role1Role recall0.20
H-bond same residue1Residue recall0.20

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
3129 5.30553003506395 -0.954123 -26.6523 3 17 17 0.85 0.40 - no Open
3167 6.173291032914957 -0.682302 -19.513 2 17 0 0.00 0.00 - no Open
3124 6.215417197943953 -0.861558 -23.485 3 18 17 0.85 0.20 - no Open
3666 6.246697130747643 -0.707757 -20.5324 6 14 0 0.00 0.00 - no Open
3670 6.272432463998912 -0.845636 -25.0388 8 14 0 0.00 0.00 - no Open
3669 6.322932638041371 -0.748965 -21.3557 4 16 0 0.00 0.00 - no Open
3668 6.6598710599952575 -0.849058 -23.1853 6 15 0 0.00 0.00 - no Open
3665 6.025346247140044 -0.740679 -21.9125 3 16 0 0.00 0.00 - yes Open
3667 6.7566606423586 -0.754286 -22.124 2 16 0 0.00 0.00 - yes Open
3126 7.2101202371091855 -0.859099 -23.8735 5 18 17 0.85 0.40 - yes Open
3127 8.241268674929234 -0.810159 -23.3605 4 18 17 0.85 0.20 - yes Open
3166 9.2308098260559 -0.854714 -23.6189 3 20 0 0.00 0.00 - yes Open
3125 9.317699948251644 -0.863629 -23.5269 2 18 15 0.75 0.20 - yes Open
3128 10.682020037457598 -0.875906 -22.7817 4 13 10 0.50 0.20 - yes Current

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -22.782kcal/mol
Ligand efficiency (LE) -0.7594kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -7.325
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 30HA

Physicochemical properties

Molecular weight 420.9Da
Lipinski: ≤ 500 Da
LogP (cLogP) 3.94
Lipinski: ≤ 5
Rotatable bonds 5

Conformational strain (MMFF94s)

Strain energy (ΔE) 26.15kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 72.32kcal/mol
Minimised FF energy 46.17kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.