FAIRMol

Z56784540

Pose ID 6333 Compound 599 Pose 3015

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Excellent LE (-0.671 kcal/mol/HA) ✓ Good fit quality (FQ -6.71) ✗ Very high strain energy (22.6 kcal/mol) ✗ Geometry warnings ✗ Protein contact clashes ℹ SASA not computed
Score
-22.812
kcal/mol
LE
-0.671
kcal/mol/HA
Fit Quality
-6.71
FQ (Leeson)
HAC
34
heavy atoms
MW
467
Da
LogP
4.87
cLogP
Strain ΔE
22.6 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, protein contact clashes, strain 22.6 kcal/mol

Interaction summary

Collapsible panels
H-bonds 1 Hydrophobic 24 π–π 4 Clashes 10 Severe clashes 0
Final rank6.1143422407634285Score-22.8118
Inter norm-0.81945Intra norm0.148516
Top1000noExcludedno
Contacts19H-bonds1
Artifact reasongeometry warning; 16 clashes; 10 protein contact clashes; high strain Δ 24.6
ResiduesA:ALA32;A:ARG48;A:ARG97;A:ASP52;A:ILE45;A:LEU94;A:LYS57;A:MET53;A:NDP301;A:PHE56;A:PHE91;A:PRO88;A:TRP47;A:TYR162;A:VAL156;A:VAL30;A:VAL31;A:VAL49;A:VAL87

Protein summary

225 residues
Protein targetT03Atoms3428
Residues225Chains2
Residue summaryLEU:380; ARG:360; VAL:272; LYS:264; ALA:240; GLU:240; PRO:224; PHE:180; THR:154; ILE:152; SER:132; TYR:126; GLN:119; ASN:98; GLY:84; NDP:74

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name3CL9Contacts20
PoseOpen native poseH-bonds9
IFP residuesA:ALA32; A:ARG97; A:ASP52; A:ILE45; A:LEU94; A:LYS57; A:MET53; A:NDP301; A:PHE56; A:PHE91; A:PRO88; A:SER86; A:THR180; A:THR54; A:THR83; A:TYR162; A:VAL156; A:VAL30; A:VAL31; A:VAL87
Current overlap16Native recall0.80
Jaccard0.70RMSD-
H-bond strict1Strict recall0.14
H-bond same residue+role1Role recall0.20
H-bond same residue1Residue recall0.20

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
2035 4.694081126021725 -0.855682 -27.5085 6 11 0 0.00 0.00 - no Open
3016 4.801540287545092 -0.956391 -29.4261 2 18 15 0.75 0.20 - no Open
3591 5.715464238322772 -0.722138 -23.6414 5 15 0 0.00 0.00 - no Open
3595 6.000774929839941 -0.738045 -20.0611 7 19 0 0.00 0.00 - no Open
3015 6.1143422407634285 -0.81945 -22.8118 1 19 16 0.80 0.20 - no Current
3596 6.30265587682257 -0.750662 -23.3545 6 17 0 0.00 0.00 - no Open
3589 6.392303134329996 -0.76255 -22.5484 4 16 0 0.00 0.00 - no Open
1988 8.237308438236917 -0.827627 -26.681 2 18 0 0.00 0.00 - no Open
2033 6.01018580957263 -0.796699 -26.1676 3 17 0 0.00 0.00 - yes Open
3592 6.461756773303042 -0.621306 -21.9507 4 17 0 0.00 0.00 - yes Open
1987 6.5407435082135645 -0.871806 -20.6974 0 15 0 0.00 0.00 - yes Open
2036 6.623910558534379 -0.986887 -31.8198 2 13 0 0.00 0.00 - yes Open
3019 6.695120878645682 -0.786034 -29.4525 0 20 19 0.95 0.00 - yes Open
1993 6.852867089436183 -0.798602 -25.7871 3 13 0 0.00 0.00 - yes Open
3014 6.853072820427299 -0.71665 -21.161 0 18 14 0.70 0.00 - yes Open
1990 6.907840345025812 -0.802543 -29.0538 4 19 0 0.00 0.00 - yes Open
1986 7.101209176856625 -0.733236 -23.0684 1 17 0 0.00 0.00 - yes Open
3018 7.892649470627741 -0.822823 -23.7287 3 14 12 0.60 0.20 - yes Open
3020 8.446452902340368 -0.793438 -21.1043 2 16 14 0.70 0.20 - yes Open
3594 9.70957943150095 -0.805989 -29.2608 7 15 0 0.00 0.00 - yes Open
1991 10.242089708916698 -0.946124 -29.5206 0 16 0 0.00 0.00 - yes Open
2034 55.992078554261276 -0.840925 -26.9181 3 18 0 0.00 0.00 - yes Open
1989 56.996523392442064 -0.883629 -31.2472 1 17 0 0.00 0.00 - yes Open
3021 57.456781196342696 -0.798441 -27.8792 3 16 14 0.70 0.20 - yes Open
3593 58.56192729339746 -0.741251 -22.7497 5 15 0 0.00 0.00 - yes Open
3017 59.19287817918776 -0.810399 -24.7281 4 13 9 0.45 0.20 - yes Open
3590 59.504999651110296 -0.699695 -19.8092 5 15 0 0.00 0.00 - yes Open
1992 60.7587420827621 -0.869064 -24.2589 3 20 0 0.00 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -22.812kcal/mol
Ligand efficiency (LE) -0.6709kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -6.713
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 34HA

Physicochemical properties

Molecular weight 466.6Da
Lipinski: ≤ 500 Da
LogP (cLogP) 4.87
Lipinski: ≤ 5
Rotatable bonds 7

Conformational strain (MMFF94s)

Strain energy (ΔE) 22.63kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 105.07kcal/mol
Minimised FF energy 82.44kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.