FAIRMol

Z71577027

Pose ID 5978 Compound 606 Pose 2660

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Excellent LE (-0.733 kcal/mol/HA) ✓ Good fit quality (FQ -6.75) ✓ Good H-bonds (3 bonds) ✗ Very high strain energy (25.6 kcal/mol) ✗ Geometry warnings ℹ SASA not computed
Score
-19.044
kcal/mol
LE
-0.733
kcal/mol/HA
Fit Quality
-6.75
FQ (Leeson)
HAC
26
heavy atoms
MW
369
Da
LogP
2.84
cLogP
Strain ΔE
25.6 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, strain 25.6 kcal/mol

Interaction summary

Collapsible panels
H-bonds 3 Hydrophobic 24 π–π 3 Clashes 12 Severe clashes 2
Final rank9.3396848045856Score-19.044
Inter norm-1.06417Intra norm0.331708
Top1000noExcludedyes
Contacts15H-bonds3
Artifact reasonexcluded; geometry warning; 11 clashes; 2 protein clashes; high strain Δ 42.8
ResiduesA:ALA32;A:ARG97;A:ASP52;A:ILE45;A:LEU94;A:LYS57;A:LYS95;A:MET53;A:NDP301;A:PHE56;A:PHE91;A:PRO93;A:THR180;A:VAL30;A:VAL31

Protein summary

225 residues
Protein targetT03Atoms3428
Residues225Chains2
Residue summaryLEU:380; ARG:360; VAL:272; LYS:264; ALA:240; GLU:240; PRO:224; PHE:180; THR:154; ILE:152; SER:132; TYR:126; GLN:119; ASN:98; GLY:84; NDP:74

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name3CL9Contacts20
PoseOpen native poseH-bonds9
IFP residuesA:ALA32; A:ARG97; A:ASP52; A:ILE45; A:LEU94; A:LYS57; A:MET53; A:NDP301; A:PHE56; A:PHE91; A:PRO88; A:SER86; A:THR180; A:THR54; A:THR83; A:TYR162; A:VAL156; A:VAL30; A:VAL31; A:VAL87
Current overlap13Native recall0.65
Jaccard0.59RMSD-
H-bond strict2Strict recall0.29
H-bond same residue+role1Role recall0.20
H-bond same residue1Residue recall0.20

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
1194 3.3330933994231584 -0.775569 -19.1656 1 13 0 0.00 0.00 - no Open
2066 3.746020292766851 -0.688109 -21.0053 6 12 0 0.00 0.00 - no Open
1196 4.080938656014805 -0.804298 -19.9796 2 12 0 0.00 0.00 - no Open
1193 4.225282388448564 -0.767966 -18.7252 1 12 0 0.00 0.00 - no Open
1816 4.403569138286684 -0.745802 -21.369 4 15 0 0.00 0.00 - no Open
1195 4.815807510469393 -0.904031 -24.7577 1 12 0 0.00 0.00 - no Open
2663 4.899918197049692 -0.931164 -21.721 2 16 16 0.80 0.20 - no Open
1819 5.587276140508173 -0.583483 -15.0875 7 14 0 0.00 0.00 - no Open
1593 5.632498254449315 -0.814464 -19.6799 2 15 0 0.00 0.00 - no Open
1243 6.596835662525375 -0.916955 -21.2025 3 16 1 0.05 0.00 - no Open
2068 6.253660736156609 -0.672619 -20.433 6 9 0 0.00 0.00 - yes Open
2069 6.284650086704847 -0.660892 -16.0336 6 9 0 0.00 0.00 - yes Open
2070 6.98568342562347 -0.672115 -14.0837 7 8 0 0.00 0.00 - yes Open
1592 7.182700776310237 -0.813693 -23.6292 2 15 0 0.00 0.00 - yes Open
1817 7.525975222622855 -0.718907 -18.6129 6 14 0 0.00 0.00 - yes Open
2661 7.551928228801605 -0.785766 -19.2447 2 15 13 0.65 0.20 - yes Open
1242 7.63896418141783 -0.913808 -22.9851 3 16 1 0.05 0.00 - yes Open
1245 8.791171282926179 -0.729578 -18.3048 6 15 1 0.05 0.00 - yes Open
2067 8.9829338433256 -0.649697 -11.3924 6 11 0 0.00 0.00 - yes Open
1818 9.198691320721796 -0.824987 -18.7544 9 14 0 0.00 0.00 - yes Open
2660 9.3396848045856 -1.06417 -19.044 3 15 13 0.65 0.20 - yes Current
2662 9.370883843603515 -0.920609 -20.4658 3 14 13 0.65 0.20 - yes Open
1244 9.933492211023694 -0.753887 -19.6855 5 14 1 0.05 0.00 - yes Open
1591 10.198157148767574 -0.847332 -20.3988 2 15 0 0.00 0.00 - yes Open
1590 11.88924984012254 -0.933543 -22.4803 6 15 0 0.00 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -19.044kcal/mol
Ligand efficiency (LE) -0.7325kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -6.748
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 26HA

Physicochemical properties

Molecular weight 369.4Da
Lipinski: ≤ 500 Da
LogP (cLogP) 2.84
Lipinski: ≤ 5
Rotatable bonds 5

Conformational strain (MMFF94s)

Strain energy (ΔE) 25.60kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 57.89kcal/mol
Minimised FF energy 32.29kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.