FAIRMol

Z49605060

Pose ID 5758 Compound 626 Pose 2440

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Excellent LE (-0.420 kcal/mol/HA) ✓ Good fit quality (FQ -3.92) ✓ Good H-bonds (3 bonds) ✗ Very high strain energy (25.4 kcal/mol) ✗ Geometry warnings ℹ SASA not computed
Score
-11.344
kcal/mol
LE
-0.420
kcal/mol/HA
Fit Quality
-3.92
FQ (Leeson)
HAC
27
heavy atoms
MW
389
Da
LogP
1.65
cLogP
Strain ΔE
25.4 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, strain 25.4 kcal/mol

Interaction summary

Collapsible panels
H-bonds 3 Hydrophobic 21 π–π 1 Clashes 19 Severe clashes 5
Final rank13.20656383768732Score-11.3443
Inter norm-0.780294Intra norm0.360135
Top1000noExcludedyes
Contacts14H-bonds3
Artifact reasonexcluded; geometry warning; 6 clashes; 5 protein clashes; high strain Δ 31.8
ResiduesA:ARG97;A:ILE45;A:LEU94;A:LYS57;A:LYS95;A:MET53;A:NDP301;A:PHE56;A:PHE91;A:PRO88;A:PRO93;A:SER44;A:SER86;A:VAL87

Protein summary

225 residues
Protein targetT03Atoms3428
Residues225Chains2
Residue summaryLEU:380; ARG:360; VAL:272; LYS:264; ALA:240; GLU:240; PRO:224; PHE:180; THR:154; ILE:152; SER:132; TYR:126; GLN:119; ASN:98; GLY:84; NDP:74

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name3CL9Contacts20
PoseOpen native poseH-bonds9
IFP residuesA:ALA32; A:ARG97; A:ASP52; A:ILE45; A:LEU94; A:LYS57; A:MET53; A:NDP301; A:PHE56; A:PHE91; A:PRO88; A:SER86; A:THR180; A:THR54; A:THR83; A:TYR162; A:VAL156; A:VAL30; A:VAL31; A:VAL87
Current overlap11Native recall0.55
Jaccard0.48RMSD-
H-bond strict1Strict recall0.14
H-bond same residue+role1Role recall0.20
H-bond same residue1Residue recall0.20

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
1369 4.2067414667746466 -0.981867 -22.6681 9 18 0 0.00 0.00 - no Open
1819 4.7572323917008195 -0.744168 -24.2371 5 9 0 0.00 0.00 - no Open
2437 5.147898269033301 -1.06094 -32.6346 3 14 13 0.65 0.40 - no Open
979 5.73744667772116 -1.13132 -30.8731 11 18 0 0.00 0.00 - no Open
1825 6.130601681038156 -0.61434 -21.0053 7 10 0 0.00 0.00 - no Open
1823 5.035408152499395 -0.678869 -19.9772 5 11 0 0.00 0.00 - yes Open
1822 5.5745355184588465 -0.739879 -17.8444 8 12 0 0.00 0.00 - yes Open
1816 5.673900758652186 -0.850416 -19.456 12 11 0 0.00 0.00 - yes Open
2442 6.0486424804734735 -0.794932 -19.5034 4 14 12 0.60 0.00 - yes Open
2436 6.127180061691416 -0.940266 -24.6331 3 16 14 0.70 0.00 - yes Open
2434 6.130982708603371 -0.829458 -17.1175 4 15 13 0.65 0.00 - yes Open
1820 6.173831864554822 -0.657543 -13.7134 8 10 0 0.00 0.00 - yes Open
983 6.319641516149942 -0.996616 -25.4921 3 15 0 0.00 0.00 - yes Open
2443 6.464614519025771 -0.969669 -32.2107 8 12 11 0.55 0.40 - yes Open
1817 6.549370517071881 -0.789605 -19.8353 8 10 0 0.00 0.00 - yes Open
1824 6.699420394745864 -0.514093 -17.8951 4 8 0 0.00 0.00 - yes Open
1818 6.783012465613875 -0.649106 -21.28 3 10 0 0.00 0.00 - yes Open
1376 7.113811811465945 -0.959319 -23.7154 10 13 0 0.00 0.00 - yes Open
1372 7.211360022403535 -0.89247 -24.2441 8 12 0 0.00 0.00 - yes Open
1368 7.3063578494846135 -0.979595 -20.8298 9 13 0 0.00 0.00 - yes Open
1821 7.420027589188007 -0.594101 -14.529 6 9 0 0.00 0.00 - yes Open
2435 7.433017776140588 -0.987052 -20.1565 5 17 16 0.80 0.60 - yes Open
1377 7.682433258561182 -0.97278 -26.5689 12 18 0 0.00 0.00 - yes Open
981 7.76045287915965 -0.901826 -23.0267 5 15 0 0.00 0.00 - yes Open
1370 7.7814666906879495 -0.986431 -27.245 10 14 0 0.00 0.00 - yes Open
1371 8.762274222805406 -0.955723 -25.8073 11 18 0 0.00 0.00 - yes Open
1375 9.068434884376416 -1.01379 -23.0943 6 18 0 0.00 0.00 - yes Open
2439 9.143238928302978 -0.917732 -24.6649 6 12 9 0.45 0.20 - yes Open
2441 9.68307304315479 -0.956771 -26.8399 5 16 14 0.70 0.40 - yes Open
2438 9.901200860898207 -0.809611 -19.3279 3 13 9 0.45 0.20 - yes Open
985 10.020070098757985 -1.18816 -36.955 6 14 0 0.00 0.00 - yes Open
977 11.177438893279382 -1.28056 -31.9367 8 14 0 0.00 0.00 - yes Open
984 11.19428606701474 -1.02116 -31.9133 6 13 0 0.00 0.00 - yes Open
1373 11.403952809413063 -1.03551 -21.5961 9 18 0 0.00 0.00 - yes Open
1374 11.46718422832834 -0.827428 -17.3766 11 19 0 0.00 0.00 - yes Open
980 12.965540698242858 -1.15396 -25.8128 6 19 0 0.00 0.00 - yes Open
2440 13.20656383768732 -0.780294 -11.3443 3 14 11 0.55 0.20 - yes Current
976 14.05385730983681 -1.27503 -27.6545 6 21 0 0.00 0.00 - yes Open
978 15.182778967909266 -1.0563 -29.3728 9 19 0 0.00 0.00 - yes Open
982 15.325270646122474 -0.955161 -20.4247 6 19 0 0.00 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -11.344kcal/mol
Ligand efficiency (LE) -0.4202kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -3.920
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 27HA

Physicochemical properties

Molecular weight 389.4Da
Lipinski: ≤ 500 Da
LogP (cLogP) 1.65
Lipinski: ≤ 5
Rotatable bonds 5

Conformational strain (MMFF94s)

Strain energy (ΔE) 25.42kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 21.43kcal/mol
Minimised FF energy -3.99kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.