FAIRMol

OSA_Lib_132

Pose ID 4470 Compound 508 Pose 1152

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Excellent LE (-0.658 kcal/mol/HA) ✓ Good fit quality (FQ -6.53) ✗ Very high strain energy (49.8 kcal/mol) ✗ Geometry warnings ✗ Protein contact clashes ℹ SASA not computed
Score
-21.728
kcal/mol
LE
-0.658
kcal/mol/HA
Fit Quality
-6.53
FQ (Leeson)
HAC
33
heavy atoms
MW
448
Da
LogP
2.62
cLogP
Strain ΔE
49.8 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, protein contact clashes, strain 49.8 kcal/mol

Interaction summary

Collapsible panels
H-bonds 1 Hydrophobic 24 π–π 2 Clashes 1 Severe clashes 0
Final rank3.615842987036019Score-21.7283
Inter norm-0.644492Intra norm-0.0139416
Top1000noExcludedno
Contacts18H-bonds1
Artifact reasongeometry warning; 12 clashes; 1 protein contact clash; high strain Δ 36.4
ResiduesA:ALA32;A:ARG48;A:ASP52;A:ILE45;A:LEU94;A:MET53;A:NDP301;A:PHE56;A:PRO88;A:SER44;A:SER86;A:TRP47;A:TYR162;A:VAL156;A:VAL30;A:VAL31;A:VAL49;A:VAL87

Protein summary

225 residues
Protein targetT03Atoms3428
Residues225Chains2
Residue summaryLEU:380; ARG:360; VAL:272; LYS:264; ALA:240; GLU:240; PRO:224; PHE:180; THR:154; ILE:152; SER:132; TYR:126; GLN:119; ASN:98; GLY:84; NDP:74

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name3CL9Contacts20
PoseOpen native poseH-bonds9
IFP residuesA:ALA32; A:ARG97; A:ASP52; A:ILE45; A:LEU94; A:LYS57; A:MET53; A:NDP301; A:PHE56; A:PHE91; A:PRO88; A:SER86; A:THR180; A:THR54; A:THR83; A:TYR162; A:VAL156; A:VAL30; A:VAL31; A:VAL87
Current overlap14Native recall0.70
Jaccard0.58RMSD-
H-bond strict0Strict recall0.00
H-bond same residue+role0Role recall0.00
H-bond same residue0Residue recall0.00

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
1152 3.615842987036019 -0.644492 -21.7283 1 18 14 0.70 0.00 - no Current
1149 4.181765261260168 -0.635062 -20.4312 0 18 15 0.75 0.00 - no Open
1151 5.165900505947793 -0.652283 -18.7734 0 16 16 0.80 0.00 - no Open
1153 54.836235310061454 -0.800754 -25.5112 0 19 17 0.85 0.00 - no Open
1155 55.028170851487445 -0.580756 -16.0531 1 18 14 0.70 0.00 - yes Open
1154 55.178575545847835 -0.664819 -16.3451 0 19 14 0.70 0.00 - yes Open
1156 56.38292227545571 -0.610732 -15.1304 0 18 14 0.70 0.00 - yes Open
1150 58.120565172577194 -0.74335 -22.7204 0 20 16 0.80 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -21.728kcal/mol
Ligand efficiency (LE) -0.6584kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -6.533
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 33HA

Physicochemical properties

Molecular weight 447.7Da
Lipinski: ≤ 500 Da
LogP (cLogP) 2.62
Lipinski: ≤ 5
Rotatable bonds 7

Conformational strain (MMFF94s)

Strain energy (ΔE) 49.82kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 177.36kcal/mol
Minimised FF energy 127.54kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.