FAIRMol

KB_chagas_92

Pose ID 3933 Compound 535 Pose 615

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Excellent LE (-0.853 kcal/mol/HA) ✓ Good fit quality (FQ -8.47) ✓ Good H-bonds (3 bonds) ✗ Very high strain energy (28.2 kcal/mol) ✗ Geometry warnings ℹ SASA not computed
Score
-28.157
kcal/mol
LE
-0.853
kcal/mol/HA
Fit Quality
-8.47
FQ (Leeson)
HAC
33
heavy atoms
MW
445
Da
LogP
0.49
cLogP
Strain ΔE
28.2 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, strain 28.2 kcal/mol

Interaction summary

Collapsible panels
H-bonds 3 Hydrophobic 24 π–π 3 Clashes 9 Severe clashes 1
Final rank6.1943138389988555Score-28.1568
Inter norm-0.890133Intra norm0.0368969
Top1000noExcludedyes
Contacts17H-bonds3
Artifact reasonexcluded; geometry warning; 10 clashes; 1 protein clash; high strain Δ 26.8
ResiduesA:ALA32;A:ARG97;A:ASP52;A:ILE45;A:LEU94;A:LYS57;A:LYS90;A:LYS95;A:MET53;A:NDP301;A:PHE56;A:PHE91;A:PRO88;A:THR180;A:VAL30;A:VAL31;A:VAL87

Protein summary

225 residues
Protein targetT03Atoms3428
Residues225Chains2
Residue summaryLEU:380; ARG:360; VAL:272; LYS:264; ALA:240; GLU:240; PRO:224; PHE:180; THR:154; ILE:152; SER:132; TYR:126; GLN:119; ASN:98; GLY:84; NDP:74

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name3CL9Contacts20
PoseOpen native poseH-bonds9
IFP residuesA:ALA32; A:ARG97; A:ASP52; A:ILE45; A:LEU94; A:LYS57; A:MET53; A:NDP301; A:PHE56; A:PHE91; A:PRO88; A:SER86; A:THR180; A:THR54; A:THR83; A:TYR162; A:VAL156; A:VAL30; A:VAL31; A:VAL87
Current overlap15Native recall0.75
Jaccard0.68RMSD-
H-bond strict2Strict recall0.29
H-bond same residue+role1Role recall0.20
H-bond same residue1Residue recall0.20

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
610 3.9227368786597183 -0.651244 -21.2159 2 15 11 0.55 0.00 - no Open
696 4.403344250181916 -0.500199 -13.5077 0 18 0 0.00 0.00 - no Open
698 5.454954305976354 -0.55846 -18.8801 5 14 0 0.00 0.00 - no Open
615 6.1943138389988555 -0.890133 -28.1568 3 17 15 0.75 0.20 - yes Current
611 10.252507299590931 -0.919278 -28.6542 4 17 14 0.70 0.20 - yes Open
614 10.366814282594296 -0.843316 -24.7097 5 14 12 0.60 0.20 - yes Open
695 11.732590774908134 -0.752914 -25.5713 6 14 0 0.00 0.00 - yes Open
697 12.23975649193952 -0.775301 -24.5546 6 14 0 0.00 0.00 - yes Open
613 12.404005164513254 -0.665891 -21.3396 3 10 7 0.35 0.20 - yes Open
612 60.661231820847455 -0.793129 -25.5679 3 13 7 0.35 0.20 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -28.157kcal/mol
Ligand efficiency (LE) -0.8532kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -8.466
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 33HA

Physicochemical properties

Molecular weight 444.6Da
Lipinski: ≤ 500 Da
LogP (cLogP) 0.49
Lipinski: ≤ 5
Rotatable bonds 8

Conformational strain (MMFF94s)

Strain energy (ΔE) 28.23kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 52.01kcal/mol
Minimised FF energy 23.78kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.