FAIRMol

KB_Leish_139

Pose ID 3891 Compound 641 Pose 573

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Excellent LE (-0.638 kcal/mol/HA) ✓ Good fit quality (FQ -6.33) ✓ Good H-bonds (3 bonds) ✗ Very high strain energy (30.1 kcal/mol) ✗ Geometry warnings ℹ SASA not computed
Score
-21.043
kcal/mol
LE
-0.638
kcal/mol/HA
Fit Quality
-6.33
FQ (Leeson)
HAC
33
heavy atoms
MW
486
Da
LogP
4.13
cLogP
Strain ΔE
30.1 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, strain 30.1 kcal/mol

Interaction summary

Collapsible panels
H-bonds 3 Hydrophobic 24 π–π 3 Clashes 7 Severe clashes 2
Final rank7.365291258555342Score-21.0427
Inter norm-0.752769Intra norm0.115111
Top1000noExcludedyes
Contacts16H-bonds3
Artifact reasonexcluded; geometry warning; 11 clashes; 2 protein clashes; high strain Δ 30.1
ResiduesA:ALA32;A:ARG48;A:ARG97;A:ASP52;A:ILE45;A:LEU94;A:LYS57;A:LYS95;A:MET53;A:NDP301;A:PHE56;A:PHE91;A:SER44;A:SER86;A:TRP47;A:VAL87

Protein summary

225 residues
Protein targetT03Atoms3428
Residues225Chains2
Residue summaryLEU:380; ARG:360; VAL:272; LYS:264; ALA:240; GLU:240; PRO:224; PHE:180; THR:154; ILE:152; SER:132; TYR:126; GLN:119; ASN:98; GLY:84; NDP:74

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name3CL9Contacts20
PoseOpen native poseH-bonds9
IFP residuesA:ALA32; A:ARG97; A:ASP52; A:ILE45; A:LEU94; A:LYS57; A:MET53; A:NDP301; A:PHE56; A:PHE91; A:PRO88; A:SER86; A:THR180; A:THR54; A:THR83; A:TYR162; A:VAL156; A:VAL30; A:VAL31; A:VAL87
Current overlap12Native recall0.60
Jaccard0.50RMSD-
H-bond strict1Strict recall0.14
H-bond same residue+role1Role recall0.20
H-bond same residue1Residue recall0.20

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
548 5.081908569193422 -0.690502 -13.1265 12 15 0 0.00 0.00 - no Open
547 5.0950710599395475 -0.555746 -13.9644 9 17 0 0.00 0.00 - no Open
545 5.105363872234837 -0.588521 -13.335 10 15 0 0.00 0.00 - no Open
572 5.431450296883614 -0.64754 -17.6195 2 16 12 0.60 0.20 - no Open
546 5.466427687060774 -0.590049 -15.2907 10 14 0 0.00 0.00 - no Open
1978 5.83503777108036 -0.706863 -15.9242 7 14 0 0.00 0.00 - no Open
528 5.952437885347036 -0.583201 -15.6926 4 18 0 0.00 0.00 - no Open
313 6.515163930159474 -0.647493 -14.6638 7 14 0 0.00 0.00 - no Open
311 6.536219478007521 -0.68128 -15.7724 7 14 0 0.00 0.00 - no Open
1980 6.57386179958214 -0.652397 -14.6786 8 14 0 0.00 0.00 - no Open
527 7.302718540145861 -0.639006 -20.2417 3 15 0 0.00 0.00 - no Open
571 6.659052124756004 -0.74966 -23.8694 3 17 16 0.80 0.20 - yes Open
525 6.751843990980415 -0.707534 -17.5975 7 13 0 0.00 0.00 - yes Open
573 7.365291258555342 -0.752769 -21.0427 3 16 12 0.60 0.20 - yes Current
526 7.604629144541703 -0.609451 -19.5701 3 13 0 0.00 0.00 - yes Open
1979 9.388373661081921 -0.70394 -14.3394 6 16 0 0.00 0.00 - yes Open
1977 9.52335982345675 -0.749603 -15.8986 7 17 0 0.00 0.00 - yes Open
574 57.26584774044052 -0.689563 -15.7303 3 17 12 0.60 0.20 - yes Open
312 59.780855866016466 -0.67002 -13.1303 10 17 0 0.00 0.00 - yes Open
310 60.46822861850252 -0.694192 -15.1833 6 15 0 0.00 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -21.043kcal/mol
Ligand efficiency (LE) -0.6377kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -6.327
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 33HA

Physicochemical properties

Molecular weight 485.6Da
Lipinski: ≤ 500 Da
LogP (cLogP) 4.13
Lipinski: ≤ 5
Rotatable bonds 7

Conformational strain (MMFF94s)

Strain energy (ΔE) 30.10kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 103.71kcal/mol
Minimised FF energy 73.61kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.