FAIRMol

KB_Leish_41

Pose ID 3848 Compound 702 Pose 530

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Excellent LE (-0.857 kcal/mol/HA) ✓ Good fit quality (FQ -8.43) ✓ Good H-bonds (5 bonds) ✗ Very high strain energy (20.2 kcal/mol) ✗ Geometry warnings ✗ Protein contact clashes ℹ SASA not computed
Score
-27.420
kcal/mol
LE
-0.857
kcal/mol/HA
Fit Quality
-8.43
FQ (Leeson)
HAC
32
heavy atoms
MW
432
Da
LogP
0.83
cLogP
Strain ΔE
20.2 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, protein contact clashes, strain 20.2 kcal/mol

Interaction summary

Collapsible panels
H-bonds 5 Hydrophobic 24 π–π 2 Clashes 11 Severe clashes 0
Final rank6.605912727722192Score-27.4202
Inter norm-0.809895Intra norm-0.0469893
Top1000noExcludedno
Contacts20H-bonds5
Artifact reasongeometry warning; 12 clashes; 11 protein contact clashes; high strain Δ 36.6
ResiduesA:ALA32;A:ASP52;A:ILE224;A:ILE45;A:LEU94;A:MET53;A:NDP301;A:PHE55;A:PHE56;A:PRO88;A:SER44;A:SER86;A:THR180;A:THR83;A:TYR162;A:TYR178;A:VAL156;A:VAL30;A:VAL31;A:VAL87

Protein summary

225 residues
Protein targetT03Atoms3428
Residues225Chains2
Residue summaryLEU:380; ARG:360; VAL:272; LYS:264; ALA:240; GLU:240; PRO:224; PHE:180; THR:154; ILE:152; SER:132; TYR:126; GLN:119; ASN:98; GLY:84; NDP:74

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name3CL9Contacts20
PoseOpen native poseH-bonds9
IFP residuesA:ALA32; A:ARG97; A:ASP52; A:ILE45; A:LEU94; A:LYS57; A:MET53; A:NDP301; A:PHE56; A:PHE91; A:PRO88; A:SER86; A:THR180; A:THR54; A:THR83; A:TYR162; A:VAL156; A:VAL30; A:VAL31; A:VAL87
Current overlap16Native recall0.80
Jaccard0.67RMSD-
H-bond strict1Strict recall0.14
H-bond same residue+role1Role recall0.20
H-bond same residue1Residue recall0.20

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
491 4.918248685407759 -0.937426 -26.6984 5 21 1 0.05 0.00 - no Open
595 5.575090899916919 -0.7408 -24.8635 4 18 0 0.00 0.00 - no Open
414 6.434035714449353 -0.717975 -25.5926 4 13 1 0.05 0.00 - no Open
485 6.500526567711173 -0.675873 -24.2658 4 13 0 0.00 0.00 - no Open
530 6.605912727722192 -0.809895 -27.4202 5 20 16 0.80 0.20 - no Current
484 7.658521530819854 -0.628344 -18.6935 2 13 0 0.00 0.00 - yes Open
529 8.323509071516625 -0.964933 -23.9292 7 20 16 0.80 0.20 - yes Open
490 8.55090867045927 -0.776061 -19.809 3 19 1 0.05 0.00 - yes Open
594 10.819536765416256 -0.842022 -25.106 5 19 0 0.00 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -27.420kcal/mol
Ligand efficiency (LE) -0.8569kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -8.427
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 32HA

Physicochemical properties

Molecular weight 431.5Da
Lipinski: ≤ 500 Da
LogP (cLogP) 0.83
Lipinski: ≤ 5
Rotatable bonds 8

Conformational strain (MMFF94s)

Strain energy (ΔE) 20.18kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 84.05kcal/mol
Minimised FF energy 63.87kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.