FAIRMol

KB_HAT_151

Pose ID 3786 Compound 418 Pose 468

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Excellent LE (-0.725 kcal/mol/HA) ✓ Good fit quality (FQ -7.25) ✗ Very high strain energy (39.8 kcal/mol) ✗ Geometry warnings ✗ Protein contact clashes ℹ SASA not computed
Score
-24.637
kcal/mol
LE
-0.725
kcal/mol/HA
Fit Quality
-7.25
FQ (Leeson)
HAC
34
heavy atoms
MW
491
Da
LogP
0.68
cLogP
Strain ΔE
39.8 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, protein contact clashes, strain 39.8 kcal/mol

Interaction summary

Collapsible panels
H-bonds 1 Hydrophobic 24 π–π 2 Clashes 8 Severe clashes 0
Final rank6.827904118123914Score-24.6373
Inter norm-0.746868Intra norm0.0222419
Top1000noExcludedno
Contacts17H-bonds1
Artifact reasongeometry warning; 11 clashes; 8 protein contact clashes; high strain Δ 54.8
ResiduesA:ALA32;A:ARG97;A:ASP52;A:LEU94;A:LYS57;A:LYS95;A:MET53;A:NDP301;A:PHE56;A:PHE91;A:PRO93;A:THR83;A:TYR162;A:VAL156;A:VAL30;A:VAL31;A:VAL87

Protein summary

225 residues
Protein targetT03Atoms3428
Residues225Chains2
Residue summaryLEU:380; ARG:360; VAL:272; LYS:264; ALA:240; GLU:240; PRO:224; PHE:180; THR:154; ILE:152; SER:132; TYR:126; GLN:119; ASN:98; GLY:84; NDP:74

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name3CL9Contacts20
PoseOpen native poseH-bonds9
IFP residuesA:ALA32; A:ARG97; A:ASP52; A:ILE45; A:LEU94; A:LYS57; A:MET53; A:NDP301; A:PHE56; A:PHE91; A:PRO88; A:SER86; A:THR180; A:THR54; A:THR83; A:TYR162; A:VAL156; A:VAL30; A:VAL31; A:VAL87
Current overlap15Native recall0.75
Jaccard0.68RMSD-
H-bond strict0Strict recall0.00
H-bond same residue+role0Role recall0.00
H-bond same residue0Residue recall0.00

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
423 6.235444614885987 -0.921178 -28.5461 4 13 0 0.00 0.00 - no Open
424 6.5752281328867355 -1.00078 -28.5431 7 14 0 0.00 0.00 - no Open
468 6.827904118123914 -0.746868 -24.6373 1 17 15 0.75 0.00 - no Current
601 7.401065038593859 -0.779113 -26.4587 2 20 0 0.00 0.00 - no Open
600 6.751124317430976 -0.70137 -19.2185 4 18 0 0.00 0.00 - yes Open
602 7.494104916731109 -0.827691 -22.9203 4 18 0 0.00 0.00 - yes Open
467 8.007040405112697 -0.677413 -17.4227 1 17 16 0.80 0.00 - yes Open
420 8.66704616002394 -0.810841 -22.9533 4 16 0 0.00 0.00 - yes Open
421 9.458859204989842 -0.907133 -29.9858 3 19 0 0.00 0.00 - yes Open
422 10.017601772255048 -0.907876 -25.4826 10 16 0 0.00 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -24.637kcal/mol
Ligand efficiency (LE) -0.7246kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -7.251
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 34HA

Physicochemical properties

Molecular weight 490.6Da
Lipinski: ≤ 500 Da
LogP (cLogP) 0.68
Lipinski: ≤ 5
Rotatable bonds 7

Conformational strain (MMFF94s)

Strain energy (ΔE) 39.84kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 171.04kcal/mol
Minimised FF energy 131.20kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.