FAIRMol

OHD_TB2022_44

Pose ID 3646 Compound 461 Pose 328

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Promising Reasonable quality metrics. Warrants further investigation.
✓ Excellent LE (-1.236 kcal/mol/HA) ✓ Good fit quality (FQ -10.73) ✓ Good H-bonds (5 bonds) ✗ Moderate strain (9.4 kcal/mol) ✗ Geometry warnings ℹ SASA not computed
Score
-27.195
kcal/mol
LE
-1.236
kcal/mol/HA
Fit Quality
-10.73
FQ (Leeson)
HAC
22
heavy atoms
MW
335
Da
LogP
3.13
cLogP
Strain ΔE
9.4 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes

Interaction summary

Collapsible panels
H-bonds 5 Hydrophobic 24 π–π 1 Clashes 6 Severe clashes 1
Final rank4.296230231162304Score-27.1953
Inter norm-1.24509Intra norm0.00894173
Top1000noExcludedyes
Contacts16H-bonds5
Artifact reasonexcluded; geometry warning; 10 clashes; 1 protein clash
ResiduesA:ALA32;A:ARG48;A:ASP52;A:ILE45;A:MET53;A:NDP301;A:PHE56;A:SER44;A:THR180;A:THR83;A:TRP47;A:TYR162;A:VAL156;A:VAL30;A:VAL31;A:VAL49

Protein summary

225 residues
Protein targetT03Atoms3428
Residues225Chains2
Residue summaryLEU:380; ARG:360; VAL:272; LYS:264; ALA:240; GLU:240; PRO:224; PHE:180; THR:154; ILE:152; SER:132; TYR:126; GLN:119; ASN:98; GLY:84; NDP:74

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name3CL9Contacts20
PoseOpen native poseH-bonds9
IFP residuesA:ALA32; A:ARG97; A:ASP52; A:ILE45; A:LEU94; A:LYS57; A:MET53; A:NDP301; A:PHE56; A:PHE91; A:PRO88; A:SER86; A:THR180; A:THR54; A:THR83; A:TYR162; A:VAL156; A:VAL30; A:VAL31; A:VAL87
Current overlap12Native recall0.60
Jaccard0.50RMSD-
H-bond strict1Strict recall0.14
H-bond same residue+role1Role recall0.20
H-bond same residue1Residue recall0.20

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
258 1.9231072611769422 -1.64315 -32.5986 5 16 0 0.00 0.00 - no Open
327 2.301671752784981 -1.17511 -21.7344 9 18 14 0.70 0.80 - no Open
218 2.3062645060307396 -1.24611 -27.9192 10 18 1 0.05 0.00 - no Open
257 2.4180250549174094 -1.72565 -35.5435 8 17 0 0.00 0.00 - no Open
217 2.4674633460653235 -1.24105 -23.9131 10 17 1 0.05 0.00 - no Open
259 2.589489975519082 -1.75118 -36.1308 6 18 0 0.00 0.00 - no Open
219 3.5259849123113742 -1.18961 -26.6206 5 19 1 0.05 0.00 - no Open
326 3.4374975848591176 -1.19404 -22.6531 10 20 16 0.80 0.80 - yes Open
328 4.296230231162304 -1.24509 -27.1953 5 16 12 0.60 0.20 - yes Current

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -27.195kcal/mol
Ligand efficiency (LE) -1.2362kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -10.732
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 22HA

Physicochemical properties

Molecular weight 335.2Da
Lipinski: ≤ 500 Da
LogP (cLogP) 3.13
Lipinski: ≤ 5
Rotatable bonds 3

Conformational strain (MMFF94s)

Strain energy (ΔE) 9.37kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 19.80kcal/mol
Minimised FF energy 10.43kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.