FAIRMol

OHD_TB2020_45

Pose ID 3577 Compound 422 Pose 259

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Excellent LE (-0.548 kcal/mol/HA) ✓ Good fit quality (FQ -5.65) ✓ Good H-bonds (4 bonds) ✗ Very high strain energy (32.9 kcal/mol) ✗ Geometry warnings ✗ Protein contact clashes ℹ SASA not computed
Score
-20.826
kcal/mol
LE
-0.548
kcal/mol/HA
Fit Quality
-5.65
FQ (Leeson)
HAC
38
heavy atoms
MW
508
Da
LogP
3.22
cLogP
Strain ΔE
32.9 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, protein contact clashes, strain 32.9 kcal/mol

Interaction summary

Collapsible panels
H-bonds 4 Hydrophobic 24 π–π 2 Clashes 14 Severe clashes 0
Final rank9.088810049341534Score-20.8257
Inter norm-0.726832Intra norm0.178787
Top1000noExcludedno
Contacts20H-bonds4
Artifact reasongeometry warning; 15 clashes; 14 protein contact clashes; high strain Δ 53.2
ResiduesA:ALA32;A:ARG97;A:ASN58;A:ASP52;A:ILE45;A:LEU94;A:LYS57;A:LYS95;A:MET53;A:NDP301;A:PHE56;A:PHE91;A:PRO88;A:PRO93;A:THR54;A:TYR162;A:VAL156;A:VAL30;A:VAL31;A:VAL87

Protein summary

225 residues
Protein targetT03Atoms3428
Residues225Chains2
Residue summaryLEU:380; ARG:360; VAL:272; LYS:264; ALA:240; GLU:240; PRO:224; PHE:180; THR:154; ILE:152; SER:132; TYR:126; GLN:119; ASN:98; GLY:84; NDP:74

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name3CL9Contacts20
PoseOpen native poseH-bonds9
IFP residuesA:ALA32; A:ARG97; A:ASP52; A:ILE45; A:LEU94; A:LYS57; A:MET53; A:NDP301; A:PHE56; A:PHE91; A:PRO88; A:SER86; A:THR180; A:THR54; A:THR83; A:TYR162; A:VAL156; A:VAL30; A:VAL31; A:VAL87
Current overlap17Native recall0.85
Jaccard0.74RMSD-
H-bond strict0Strict recall0.00
H-bond same residue+role0Role recall0.00
H-bond same residue0Residue recall0.00

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
182 6.391261306295667 -0.778366 -26.9037 3 21 1 0.05 0.00 - no Open
183 7.187001608844698 -0.652513 -22.3147 2 18 1 0.05 0.00 - no Open
231 7.36650346561456 -0.49034 -14.1942 5 13 0 0.00 0.00 - no Open
162 7.417001990643968 -0.602331 -17.9519 4 16 0 0.00 0.00 - no Open
235 7.496886454145249 -0.723705 -25.3375 2 19 0 0.00 0.00 - no Open
151 7.6306842273625115 -0.545053 -16.5986 4 13 1 0.05 0.00 - no Open
259 9.088810049341534 -0.726832 -20.8257 4 20 17 0.85 0.00 - no Current
233 7.19617598799369 -0.829407 -22.8732 4 20 0 0.00 0.00 - yes Open
234 8.116618596823802 -0.645816 -20.9507 2 19 0 0.00 0.00 - yes Open
161 8.267785370753245 -0.70794 -20.7382 3 18 0 0.00 0.00 - yes Open
150 9.157961841627277 -0.55121 -19.919 3 12 1 0.05 0.00 - yes Open
232 9.466225466118743 -0.477998 -14.2517 4 13 0 0.00 0.00 - yes Open
258 10.923066530499042 -0.772335 -25.6125 4 18 14 0.70 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -20.826kcal/mol
Ligand efficiency (LE) -0.5480kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -5.650
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 38HA

Physicochemical properties

Molecular weight 507.6Da
Lipinski: ≤ 500 Da
LogP (cLogP) 3.22
Lipinski: ≤ 5
Rotatable bonds 8

Conformational strain (MMFF94s)

Strain energy (ΔE) 32.89kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 105.73kcal/mol
Minimised FF energy 72.84kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.