FAIRMol

NMT-TY0621

Pose ID 2156 Compound 251 Pose 2156

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Excellent LE (-0.861 kcal/mol/HA) ✓ Good fit quality (FQ -8.22) ✗ Very high strain energy (33.9 kcal/mol) ✗ Geometry warnings ✗ Protein contact clashes ℹ SASA not computed
Score
-24.968
kcal/mol
LE
-0.861
kcal/mol/HA
Fit Quality
-8.22
FQ (Leeson)
HAC
29
heavy atoms
MW
438
Da
LogP
2.78
cLogP
Strain ΔE
33.9 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, protein contact clashes, strain 33.9 kcal/mol

Interaction summary

Collapsible panels
H-bonds 2 Hydrophobic 23 π–π 1 Clashes 6 Severe clashes 0
Final rank5.245054044339124Score-24.9684
Inter norm-0.839966Intra norm-0.0210149
Top1000noExcludedno
Contacts18H-bonds2
Artifact reasongeometry warning; 12 clashes; 6 protein contact clashes; high strain Δ 38.9
ResiduesA:ALA10;A:ASN65;A:ASP22;A:ILE61;A:ILE8;A:LEU23;A:LEU68;A:NAP201;A:PHE32;A:PHE35;A:PRO27;A:PRO62;A:SER60;A:THR57;A:TRP25;A:TYR122;A:VAL116;A:VAL9

Protein summary

200 residues
Protein targetT02Atoms3128
Residues200Chains2
Residue summaryLYS:374; LEU:361; GLU:240; VAL:224; ARG:192; PHE:180; ILE:171; PRO:168; ASN:140; SER:132; TYR:126; GLN:119; ASP:108; MET:102; THR:98; GLY:91

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name5SD8Contacts21
PoseOpen native poseH-bonds5
IFP residuesA:ALA10; A:ASN65; A:ASP22; A:GLN36; A:GLU31; A:GLY117; A:GLY21; A:ILE61; A:ILE8; A:LEU23; A:LEU68; A:NAP201; A:PHE32; A:PHE35; A:PRO62; A:SER60; A:THR137; A:THR57; A:TYR122; A:VAL116; A:VAL9
Current overlap16Native recall0.76
Jaccard0.70RMSD-
H-bond strict1Strict recall0.20
H-bond same residue+role1Role recall0.20
H-bond same residue1Residue recall0.20

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
1442 3.4035685731313396 -0.699217 -20.3472 5 11 0 0.00 0.00 - no Open
690 4.166677631370432 -0.845357 -25.7673 0 14 0 0.00 0.00 - no Open
2154 5.079344793313566 -0.862586 -24.6089 2 19 16 0.76 0.20 - no Open
2156 5.245054044339124 -0.839966 -24.9684 2 18 16 0.76 0.20 - no Current
2882 5.29001000847853 -0.751606 -24.1947 1 16 0 0.00 0.00 - no Open
1261 5.636507202051849 -0.744188 -20.9291 9 14 0 0.00 0.00 - no Open
1113 6.731353583884042 -0.721886 -21.5775 6 14 0 0.00 0.00 - no Open
689 5.106033026370598 -0.855947 -25.5191 1 14 0 0.00 0.00 - yes Open
2153 6.31214821199589 -0.897136 -28.8563 2 21 17 0.81 0.20 - yes Open
2157 6.333224029723648 -0.926537 -24.8747 6 16 12 0.57 0.40 - yes Open
2155 6.514953289611458 -0.850221 -23.7231 1 18 16 0.76 0.00 - yes Open
1443 6.650765963609981 -0.759293 -21.2289 7 14 0 0.00 0.00 - yes Open
1114 8.21927817028735 -0.940207 -27.295 6 13 0 0.00 0.00 - yes Open
2881 8.29349690404342 -0.868419 -24.2502 5 17 0 0.00 0.00 - yes Open
1445 8.404902860284816 -0.737493 -19.9434 6 12 0 0.00 0.00 - yes Open
1112 8.923719197533764 -0.681888 -18.7626 5 18 0 0.00 0.00 - yes Open
1444 8.986734609341338 -0.679317 -16.716 6 14 0 0.00 0.00 - yes Open
1260 9.75418497111321 -0.696264 -19.6386 11 16 0 0.00 0.00 - yes Open
1446 10.208036033329622 -0.653728 -21.1612 5 12 0 0.00 0.00 - yes Open
1111 11.566036702414712 -0.780764 -20.2522 1 17 0 0.00 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -24.968kcal/mol
Ligand efficiency (LE) -0.8610kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -8.219
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 29HA

Physicochemical properties

Molecular weight 437.6Da
Lipinski: ≤ 500 Da
LogP (cLogP) 2.78
Lipinski: ≤ 5
Rotatable bonds 6

Conformational strain (MMFF94s)

Strain energy (ΔE) 33.91kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 22.48kcal/mol
Minimised FF energy -11.43kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.