FAIRMol

OSA_Lib_220

Pose ID 1412 Compound 299 Pose 1412

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Excellent LE (-0.421 kcal/mol/HA) ✓ Good fit quality (FQ -4.34) ✗ Very high strain energy (29.9 kcal/mol) ✗ Geometry warnings ℹ SASA not computed
Score
-16.015
kcal/mol
LE
-0.421
kcal/mol/HA
Fit Quality
-4.34
FQ (Leeson)
HAC
38
heavy atoms
MW
518
Da
LogP
2.31
cLogP
Strain ΔE
29.9 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, strain 29.9 kcal/mol

Interaction summary

Collapsible panels
H-bonds 2 Hydrophobic 24 π–π 2 Clashes 9 Severe clashes 1
Final rank57.63987810704703Score-16.0152
Inter norm-0.631785Intra norm0.210331
Top1000noExcludedyes
Contacts19H-bonds2
Artifact reasonexcluded; geometry warning; 20 clashes; 1 protein clash
ResiduesA:ALA10;A:ARG29;A:ASN65;A:GLN36;A:GLU31;A:ILE61;A:ILE8;A:LEU23;A:LEU28;A:LEU68;A:NAP201;A:PHE32;A:PHE35;A:PRO27;A:PRO62;A:SER60;A:THR137;A:TYR122;A:VAL9

Protein summary

200 residues
Protein targetT02Atoms3128
Residues200Chains2
Residue summaryLYS:374; LEU:361; GLU:240; VAL:224; ARG:192; PHE:180; ILE:171; PRO:168; ASN:140; SER:132; TYR:126; GLN:119; ASP:108; MET:102; THR:98; GLY:91

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name5SD8Contacts21
PoseOpen native poseH-bonds5
IFP residuesA:ALA10; A:ASN65; A:ASP22; A:GLN36; A:GLU31; A:GLY117; A:GLY21; A:ILE61; A:ILE8; A:LEU23; A:LEU68; A:NAP201; A:PHE32; A:PHE35; A:PRO62; A:SER60; A:THR137; A:THR57; A:TYR122; A:VAL116; A:VAL9
Current overlap16Native recall0.76
Jaccard0.67RMSD-
H-bond strict0Strict recall0.00
H-bond same residue+role0Role recall0.00
H-bond same residue0Residue recall0.00

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
1397 5.5121144581389245 -0.49729 -18.4874 0 20 15 0.71 0.00 - no Open
1389 5.758645763083225 -0.591002 -17.9108 1 17 14 0.67 0.20 - no Open
1401 5.782123514156501 -0.488802 -15.4969 1 18 15 0.71 0.00 - no Open
1410 5.882699960713685 -0.560414 -19.7145 2 18 14 0.67 0.20 - no Open
1394 6.189802953033694 -0.592223 -21.2282 0 21 17 0.81 0.00 - no Open
1403 6.250334845652669 -0.693149 -21.5089 1 20 16 0.76 0.00 - no Open
1408 6.483746905491712 -0.444635 -14.7476 0 17 12 0.57 0.00 - no Open
1402 56.6074390296758 -0.647695 -22.8061 0 21 17 0.81 0.00 - no Open
1391 7.759311933153264 -0.528591 -21.1458 0 19 15 0.71 0.00 - yes Open
1409 10.144445370660993 -0.524993 -5.67818 1 18 15 0.71 0.20 - yes Open
1393 56.235082461874015 -0.517477 -15.0716 1 19 17 0.81 0.00 - yes Open
1400 56.703592546027096 -0.622109 -20.9323 2 18 16 0.76 0.20 - yes Open
1396 56.88340914564929 -0.628022 -11.943 1 20 16 0.76 0.00 - yes Open
1392 56.9231047733685 -0.591893 -9.50292 0 19 17 0.81 0.00 - yes Open
1412 57.63987810704703 -0.631785 -16.0152 2 19 16 0.76 0.00 - yes Current
1390 57.6718620970341 -0.568182 -20.7913 1 20 16 0.76 0.00 - yes Open
1399 57.853099961065034 -0.662282 -22.2029 1 20 18 0.86 0.20 - yes Open
1405 57.85637543809406 -0.546574 -10.4811 1 15 12 0.57 0.20 - yes Open
1395 57.96506968857736 -0.578716 -12.7797 2 21 17 0.81 0.20 - yes Open
1404 58.80533028071535 -0.526194 -14.059 1 17 13 0.62 0.00 - yes Open
1407 58.9844005084797 -0.670354 -22.6601 1 20 18 0.86 0.20 - yes Open
1398 59.4321135345235 -0.522344 -15.3171 0 19 15 0.71 0.00 - yes Open
1406 59.67224043201641 -0.476078 -15.6987 0 18 14 0.67 0.00 - yes Open
1411 59.88856743562721 -0.62081 -18.8897 1 20 16 0.76 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -16.015kcal/mol
Ligand efficiency (LE) -0.4215kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -4.345
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 38HA

Physicochemical properties

Molecular weight 517.8Da
Lipinski: ≤ 500 Da
LogP (cLogP) 2.31
Lipinski: ≤ 5
Rotatable bonds 7

Conformational strain (MMFF94s)

Strain energy (ΔE) 29.88kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 170.03kcal/mol
Minimised FF energy 140.15kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.