FAIRMol

NMT-TY0772

Pose ID 13780 Compound 481 Pose 927

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Weak Marginal quality. Consider only alongside better-scoring alternatives.
✓ Excellent LE (-1.580 kcal/mol/HA) ✓ Good fit quality (FQ -12.95) ✓ Strong H-bond network (12 bonds) ✗ High strain energy (14.5 kcal/mol) ✗ Geometry warnings ✗ Protein contact clashes ℹ SASA not computed
Score
-30.018
kcal/mol
LE
-1.580
kcal/mol/HA
Fit Quality
-12.95
FQ (Leeson)
HAC
19
heavy atoms
MW
280
Da
LogP
0.02
cLogP
Strain ΔE
14.5 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, protein contact clashes, strain 14.5 kcal/mol

Interaction summary

Collapsible panels
H-bonds 12 Hydrophobic 19 π–π 2 Clashes 9 Severe clashes 0
Final rank2.817027839794606Score-30.0181
Inter norm-1.72753Intra norm0.147633
Top1000noExcludedno
Contacts13H-bonds12
Artifact reasongeometry warning; 6 clashes; 9 protein contact clashes; moderate strain Δ 15.8
ResiduesA:ALA96;A:ARG14;A:ASP161;A:LEU208;A:LEU209;A:MET213;A:NAP301;A:PHE97;A:PRO210;A:SER95;A:TRP221;A:TYR174;A:VAL206

Protein summary

258 residues
Protein targetT08Atoms3881
Residues258Chains2
Residue summaryLEU:437; VAL:433; ALA:361; ARG:288; ILE:266; GLU:210; LYS:198; SER:198; ASN:182; THR:154; GLN:153; PHE:140; PRO:140; TYR:126; GLY:112; HIS:103

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
NameTbPTR1_cW_6RX6_ReadyContacts19
PoseOpen native poseH-bonds6
IFP residuesA:ARG14; A:ASP161; A:CYS168; A:GLY205; A:LEU208; A:LEU209; A:LYS178; A:MET213; A:NAP301; A:PHE171; A:PHE97; A:PRO210; A:PRO99; A:SER207; A:SER95; A:TRP221; A:TYR174; A:TYR98; A:VAL206
Current overlap12Native recall0.63
Jaccard0.60RMSD-
H-bond strict4Strict recall0.67
H-bond same residue+role4Role recall0.80
H-bond same residue4Residue recall0.80

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
928 2.6662103575983664 -1.85511 -29.1252 9 15 14 0.74 0.80 - no Open
927 2.817027839794606 -1.72753 -30.0181 12 13 12 0.63 0.80 - no Current
848 2.944523796123663 -1.87039 -29.4322 9 15 14 0.74 0.80 - no Open
2268 3.1170949224775 -1.30574 -24.3182 4 14 0 0.00 0.00 - no Open
910 3.39635074445896 -1.07503 -17.9023 6 17 0 0.00 0.00 - no Open
847 3.9134046702727576 -1.74874 -30.4019 11 15 14 0.74 0.80 - no Open
2266 4.1761537048642605 -1.48177 -26.4623 10 17 0 0.00 0.00 - no Open
911 5.211462340964783 -1.17556 -21.6784 5 20 0 0.00 0.00 - yes Open
2267 5.442531889953567 -1.66307 -31.0938 9 16 0 0.00 0.00 - yes Open
912 6.8469444483002535 -1.25726 -17.7812 10 20 0 0.00 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -30.018kcal/mol
Ligand efficiency (LE) -1.5799kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -12.950
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 19HA

Physicochemical properties

Molecular weight 280.3Da
Lipinski: ≤ 500 Da
LogP (cLogP) 0.02
Lipinski: ≤ 5
Rotatable bonds 3

Conformational strain (MMFF94s)

Strain energy (ΔE) 14.51kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy -82.25kcal/mol
Minimised FF energy -96.76kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.