FAIRMol

OSA_Lib_197

Pose ID 1323 Compound 174 Pose 1323

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Weak Marginal quality. Consider only alongside better-scoring alternatives.
✓ Excellent LE (-0.658 kcal/mol/HA) ✓ Good fit quality (FQ -6.47) ✗ Very high strain energy (21.1 kcal/mol) ✗ Geometry warnings ℹ SASA not computed
Score
-21.053
kcal/mol
LE
-0.658
kcal/mol/HA
Fit Quality
-6.47
FQ (Leeson)
HAC
32
heavy atoms
MW
434
Da
LogP
3.26
cLogP
Strain ΔE
21.1 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, strain 21.1 kcal/mol

Interaction summary

Collapsible panels
H-bonds 2 Hydrophobic 24 π–π 3 Clashes 11 Severe clashes 3
Final rank59.631057968599535Score-21.0531
Inter norm-0.704799Intra norm0.0468891
Top1000noExcludedyes
Contacts20H-bonds2
Artifact reasonexcluded; geometry warning; 16 clashes; 3 protein clashes
ResiduesA:ALA10;A:ASN65;A:ASP22;A:GLN36;A:GLU31;A:GLY21;A:ILE61;A:ILE8;A:LEU23;A:LEU28;A:LEU68;A:NAP201;A:PHE32;A:PHE35;A:PRO62;A:SER60;A:TRP25;A:TYR122;A:VAL116;A:VAL9

Protein summary

200 residues
Protein targetT02Atoms3128
Residues200Chains2
Residue summaryLYS:374; LEU:361; GLU:240; VAL:224; ARG:192; PHE:180; ILE:171; PRO:168; ASN:140; SER:132; TYR:126; GLN:119; ASP:108; MET:102; THR:98; GLY:91

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name5SD8Contacts21
PoseOpen native poseH-bonds5
IFP residuesA:ALA10; A:ASN65; A:ASP22; A:GLN36; A:GLU31; A:GLY117; A:GLY21; A:ILE61; A:ILE8; A:LEU23; A:LEU68; A:NAP201; A:PHE32; A:PHE35; A:PRO62; A:SER60; A:THR137; A:THR57; A:TYR122; A:VAL116; A:VAL9
Current overlap18Native recall0.86
Jaccard0.78RMSD-
H-bond strict0Strict recall0.00
H-bond same residue+role0Role recall0.00
H-bond same residue0Residue recall0.00

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
1321 4.447365121142325 -0.510365 -12.4257 1 15 12 0.57 0.00 - no Open
1320 4.642518424132285 -0.593666 -16.1833 0 18 15 0.71 0.00 - no Open
1316 4.709779236245509 -0.575202 -18.4096 0 17 17 0.81 0.00 - no Open
1312 7.228478813679798 -0.697559 -13.4692 0 22 18 0.86 0.00 - no Open
1318 53.86795922307394 -0.61179 -19.5521 0 21 18 0.86 0.00 - no Open
1324 54.63520080120113 -0.556979 -17.0053 1 20 16 0.76 0.00 - no Open
1315 55.16648896161168 -0.754032 -22.678 1 23 19 0.90 0.00 - yes Open
1310 55.61044564829666 -0.653128 -21.3775 1 20 17 0.81 0.00 - yes Open
1309 55.76190127404837 -0.547391 -13.7111 1 19 18 0.86 0.00 - yes Open
1313 55.794413469951216 -0.753903 -17.0306 3 20 16 0.76 0.00 - yes Open
1314 56.71434976946213 -0.570066 -4.51698 1 20 19 0.90 0.00 - yes Open
1311 57.55833326861145 -0.581995 -14.6443 0 20 17 0.81 0.00 - yes Open
1317 57.881109294782945 -0.59117 -9.82728 0 20 18 0.86 0.00 - yes Open
1319 57.979457399511965 -0.623997 -18.8615 1 20 17 0.81 0.20 - yes Open
1322 58.36433800471837 -0.559556 -13.7987 1 19 18 0.86 0.00 - yes Open
1323 59.631057968599535 -0.704799 -21.0531 2 20 18 0.86 0.00 - yes Current

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -21.053kcal/mol
Ligand efficiency (LE) -0.6579kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -6.470
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 32HA

Physicochemical properties

Molecular weight 433.6Da
Lipinski: ≤ 500 Da
LogP (cLogP) 3.26
Lipinski: ≤ 5
Rotatable bonds 6

Conformational strain (MMFF94s)

Strain energy (ΔE) 21.14kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 104.59kcal/mol
Minimised FF energy 83.46kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.