FAIRMol

2WOV

Pose ID 12879 Compound 5191

DB fairmolDocking pose analysis is being read from this database.
Molecular metrics status: done
RDKit SASA-based burial metrics are cached.
SASA cached
T19
T. brucei TR (NADPH binding site) T. brucei NADPH binding site
Ligand 2WOV
PDB2WOV

3D complex viewer

Strict H-bonds Permissive H-bonds
Viewer legend
Protein receptor
Pocket residues
Cofactor context
Docked ligand
Overall assessment
Reject SASA cached
Likely artefact or unreliable pose
Binding weak Geometry low Native strong SASA done
Strain ΔE
101.2 kcal/mol
Protein clashes
1
Internal clashes
24
Native overlap
contact recall 1.00, Jaccard 1.00, H-bond role recall 1.00
Burial
0%
Hydrophobic fit
0%
Reason: 24 severe internal clashes, 24 internal clashes, strain 101.2 kcal/mol
strain ΔE 101.2 kcal/mol 24 severe internal clashes 1 protein-contact clashes 24 intramolecular clashes weak burial (0% buried)
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Strong H-bond network (16 bonds) ✗ Extreme strain energy (101.2 kcal/mol) ✗ Poor burial (0% SASA buried)
HAC
48
heavy atoms
MW
741
Da
LogP
-0.82
cLogP
Strain ΔE
101.2 kcal/mol
SASA buried
0%
Lipo contact
0% BSA apolar/total
SASA unbound
958 Ų
Apolar buried
301 Ų

Interaction summary

HB 16 HY 18 PI 0 CLASH 24 Severe 24

HB · H-bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

PI · π–π interactions

No pi · π–π interactions detected for this pose.

HY · Hydrophobic contacts

CLASH · Clashes

Final rank-Score-
Inter norm-Intra norm-
Top1000noExcludedno
Contacts27H-bonds16
Artifact reasonNative reference ligand
Residues
ALA284 ALA365 ARG222 ARG228 ARG287 ASN223 ASN254 GLN165 GLU202 GLY195 GLY196 GLY197 GLY286 ILE199 ILE285 LEU227 LEU334 LYS60 MET333 NDP800 PHE198 PHE367 PRO167 SER200 TYR221 VAL194 VAL366

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name2WOVContacts27
PoseOpen native poseHB0
IFP residues
ALA284 ALA365 ARG222 ARG228 ARG287 ASN223 ASN254 GLN165 GLU202 GLY195 GLY196 GLY197 GLY286 ILE199 ILE285 LEU227 LEU334 LYS60 MET333 NDP800 PHE198 PHE367 PRO167 SER200 TYR221 VAL194 VAL366
Current overlap27Native recall1.00
Jaccard1.00RMSD0.00 Å
HB strict12Strict recall1.00
HB same residue+role5HB role recall1.00
HB same residue4HB residue recall1.00

Protein summary

493 residues
Protein targetT19Atoms7541
Residues493Chains1
Residue summaryVAL:768; LYS:704; LEU:703; ILE:532; GLU:450; THR:434; ARG:408; PHE:400; ALA:390; ASN:350; PRO:350; GLY:336; SER:330; TYR:294; ASP:264; MET:221

Receptor context

1 kept / 0 excluded
Receptor context filtering: interactions and SASA are computed against protein atoms plus allowed cofactors/ions. Native ligand-like HETATM partners are excluded from scoring.
Kept context 1 Excluded HETATM 0
Kept cofactors / ions
C:NDP800

All stored poses for this docking hit

PoseFinal rankInter normScoreHBCTCT overlapCT recallHB role rec.RMSDExcluded
- ★ Native - - - 16 27 27 1.00 1.00 0.00 Å no Current

Molecular metrics

RDKit SASA burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Heavy atom count 48HA

Physicochemical properties

Molecular weight 741.4Da
Lipinski: ≤ 500 Da
LogP (cLogP) -0.82
Lipinski: ≤ 5
Rotatable bonds 17

Conformational strain (MMFF94s)

Strain energy (ΔE) 101.24kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 70.89kcal/mol
Minimised FF energy -30.36kcal/mol

SASA & burial

✓ computed
SASA (unbound) 958.3Ų
Total solvent-accessible surface area of free ligand
BSA total 0.0Ų
Buried surface area upon binding
BSA apolar 300.9Ų
Hydrophobic contacts buried
BSA polar 227.5Ų
Polar contacts buried
Fraction buried 0.0%
> 60 % indicates good pocket engagement
Lipophilic contact ratio 0.0%
BSA apolar / BSA total — high = hydrophobic driver
Δ Non-polar SASA -2685.9Ų
SASA_nonpolar(complex) − SASA_nonpolar(receptor) − SASA_nonpolar(ligand free). Negative = non-polar surface buried upon binding. Requires full polarity-decomposed SASA computation.
Receptor non-polar SASA 4064.7Ų
Non-polar SASA of receptor alone (VdW proxy, nonpolar atoms only)
Complex non-polar SASA 1843.3Ų
Non-polar SASA of full complex (VdW proxy, nonpolar atoms only)