FAIRMol

OSA_Lib_82

Pose ID 1082 Compound 297 Pose 1082

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Good LE (-0.397 kcal/mol/HA) ✓ Good fit quality (FQ -4.07) ✓ Good H-bonds (4 bonds) ✗ Very high strain energy (35.0 kcal/mol) ✗ Geometry warnings ℹ SASA not computed
Score
-14.689
kcal/mol
LE
-0.397
kcal/mol/HA
Fit Quality
-4.07
FQ (Leeson)
HAC
37
heavy atoms
MW
505
Da
LogP
2.13
cLogP
Strain ΔE
35.0 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, strain 35.0 kcal/mol

Interaction summary

Collapsible panels
H-bonds 4 Hydrophobic 24 π–π 1 Clashes 16 Severe clashes 2
Final rank60.16059117578904Score-14.6894
Inter norm-0.566636Intra norm0.169625
Top1000noExcludedyes
Contacts20H-bonds4
Artifact reasonexcluded; geometry warning; 16 clashes; 2 protein clashes
ResiduesA:ALA10;A:ASN65;A:ASP22;A:GLU31;A:GLY21;A:ILE61;A:ILE8;A:LEU23;A:LEU28;A:LEU68;A:NAP201;A:PHE32;A:PHE35;A:PRO27;A:PRO62;A:SER60;A:TRP25;A:TYR122;A:VAL116;A:VAL9

Protein summary

200 residues
Protein targetT02Atoms3128
Residues200Chains2
Residue summaryLYS:374; LEU:361; GLU:240; VAL:224; ARG:192; PHE:180; ILE:171; PRO:168; ASN:140; SER:132; TYR:126; GLN:119; ASP:108; MET:102; THR:98; GLY:91

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name5SD8Contacts21
PoseOpen native poseH-bonds5
IFP residuesA:ALA10; A:ASN65; A:ASP22; A:GLN36; A:GLU31; A:GLY117; A:GLY21; A:ILE61; A:ILE8; A:LEU23; A:LEU68; A:NAP201; A:PHE32; A:PHE35; A:PRO62; A:SER60; A:THR137; A:THR57; A:TYR122; A:VAL116; A:VAL9
Current overlap17Native recall0.81
Jaccard0.71RMSD-
H-bond strict3Strict recall0.60
H-bond same residue+role3Role recall0.60
H-bond same residue3Residue recall0.60

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
1088 5.49466491095866 -0.602602 -21.5317 4 18 15 0.71 0.40 - no Open
1089 5.910404916945135 -0.598275 -18.5514 2 19 17 0.81 0.20 - no Open
1087 6.381627342090313 -0.613124 -19.0255 1 21 18 0.86 0.20 - no Open
1079 6.399941883630168 -0.596054 -23.2991 1 21 18 0.86 0.00 - no Open
1074 6.468691749711437 -0.620364 -17.7277 2 17 14 0.67 0.40 - no Open
1073 6.642473605057647 -0.543382 -15.5042 1 19 14 0.67 0.00 - no Open
1090 55.4106348521436 -0.674344 -24.5837 1 21 17 0.81 0.00 - no Open
1070 55.95586081193009 -0.560027 -14.7058 4 19 15 0.71 0.20 - no Open
1072 55.755462172695275 -0.54056 -18.6733 3 18 15 0.71 0.20 - yes Open
1069 55.87664166758715 -0.600282 -17.9904 1 19 16 0.76 0.20 - yes Open
1080 56.26636751020345 -0.527855 -16.0734 1 17 14 0.67 0.20 - yes Open
1084 56.47178597754696 -0.698401 -12.1278 2 20 16 0.76 0.00 - yes Open
1076 57.527861245199674 -0.7254 -12.8303 3 20 16 0.76 0.00 - yes Open
1083 57.71618768770753 -0.722603 -14.587 3 19 16 0.76 0.00 - yes Open
1071 57.73381680735157 -0.699491 -20.3995 5 17 13 0.62 0.20 - yes Open
1085 58.005416666395085 -0.591381 -17.5832 2 18 17 0.81 0.40 - yes Open
1091 58.025874117317585 -0.759207 -22.985 3 19 15 0.71 0.00 - yes Open
1078 58.10172945062032 -0.566347 -19.9464 5 18 15 0.71 0.60 - yes Open
1092 58.262648979570756 -0.760053 -19.6001 3 21 17 0.81 0.00 - yes Open
1075 58.4142773127317 -0.583239 -17.2797 2 19 16 0.76 0.40 - yes Open
1081 58.88130103939538 -0.569601 -19.2584 4 17 14 0.67 0.40 - yes Open
1077 58.938185723760796 -0.609064 -20.3775 3 20 15 0.71 0.40 - yes Open
1082 60.16059117578904 -0.566636 -14.6894 4 20 17 0.81 0.60 - yes Current
1086 60.19062111512856 -0.575684 -23.0285 0 19 16 0.76 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -14.689kcal/mol
Ligand efficiency (LE) -0.3970kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -4.065
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 37HA

Physicochemical properties

Molecular weight 504.7Da
Lipinski: ≤ 500 Da
LogP (cLogP) 2.13
Lipinski: ≤ 5
Rotatable bonds 7

Conformational strain (MMFF94s)

Strain energy (ΔE) 35.05kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 75.10kcal/mol
Minimised FF energy 40.06kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.