FAIRMol

Z56821211

Pose ID 10277 Compound 1207 Pose 1698

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Weak Marginal quality. Consider only alongside better-scoring alternatives.
✓ Excellent LE (-0.791 kcal/mol/HA) ✓ Good fit quality (FQ -7.19) ✗ High strain energy (17.1 kcal/mol) ✗ Geometry warnings ℹ SASA not computed
Score
-19.778
kcal/mol
LE
-0.791
kcal/mol/HA
Fit Quality
-7.19
FQ (Leeson)
HAC
25
heavy atoms
MW
356
Da
LogP
2.23
cLogP
Strain ΔE
17.1 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: mixed
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, strain 17.1 kcal/mol

Interaction summary

Collapsible panels
H-bonds 2 Hydrophobic 24 π–π 2 Clashes 9 Severe clashes 2
Final rank6.978943285099711Score-19.7782
Inter norm-0.809757Intra norm0.0186261
Top1000noExcludedyes
Contacts16H-bonds2
Artifact reasonexcluded; geometry warning; 8 clashes; 2 protein clashes; high strain Δ 23.9
ResiduesA:ALA34;A:ARG100;A:ARG59;A:ASP54;A:GLN56;A:GLU50;A:ILE160;A:ILE47;A:LEU97;A:MET55;A:NDP301;A:PHE58;A:PHE94;A:PRO52;A:VAL32;A:VAL33

Protein summary

223 residues
Protein targetT06Atoms3452
Residues223Chains1
Residue summaryARG:408; VAL:352; LYS:308; LEU:304; PRO:238; ILE:209; GLU:195; THR:182; SER:176; ALA:160; PHE:140; ASN:126; GLY:126; ASP:108; GLN:85; NDP:74

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name8RHTContacts21
PoseOpen native poseH-bonds6
IFP residuesA:ALA34; A:ASP54; A:HIS182; A:ILE160; A:ILE47; A:LEU90; A:LEU97; A:MET55; A:NDP301; A:PHE233; A:PHE58; A:PHE94; A:PRO91; A:SER89; A:THR184; A:THR86; A:TRP49; A:TYR166; A:TYR57; A:VAL32; A:VAL33
Current overlap11Native recall0.52
Jaccard0.42RMSD-
H-bond strict0Strict recall0.00
H-bond same residue+role0Role recall0.00
H-bond same residue0Residue recall0.00

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
2311 3.1160178135448215 -0.886933 -22.6426 7 16 0 0.00 0.00 - no Open
2266 3.3009109990344334 -0.771742 -20.5284 1 16 0 0.00 0.00 - no Open
2259 3.492922341685937 -1.01448 -23.3759 5 16 0 0.00 0.00 - no Open
2161 3.777153167833981 -1.22625 -32.2234 6 12 0 0.00 0.00 - no Open
2156 4.318860691653812 -1.10504 -24.376 10 16 0 0.00 0.00 - no Open
2160 4.322382833842899 -0.93102 -23.8202 3 10 0 0.00 0.00 - no Open
2697 4.344710715062578 -0.730464 -17.6431 6 9 0 0.00 0.00 - no Open
2305 4.470993821215696 -0.99533 -23.013 7 18 0 0.00 0.00 - no Open
2859 4.879978694211175 -0.880396 -23.2077 8 14 0 0.00 0.00 - no Open
2850 5.0745845199948105 -0.982715 -23.1512 7 17 0 0.00 0.00 - no Open
2158 5.299620021190572 -1.06324 -26.2372 4 11 0 0.00 0.00 - no Open
1696 5.734600080634052 -0.887602 -21.1051 8 18 16 0.76 1.00 - no Open
2263 6.083585839561213 -0.878106 -20.4949 6 18 0 0.00 0.00 - no Open
2262 7.307116047334361 -0.863164 -17.675 7 14 0 0.00 0.00 - no Open
2310 4.597825653045845 -0.989786 -22.1634 12 18 0 0.00 0.00 - yes Open
1693 4.634466718800378 -0.86528 -21.1269 0 17 15 0.71 0.00 - yes Open
1694 4.941961333195032 -0.854215 -18.6867 4 17 14 0.67 0.25 - yes Open
2255 5.063279742676437 -1.1021 -24.3015 6 20 0 0.00 0.00 - yes Open
2848 5.116912139779588 -0.947626 -21.9115 5 16 0 0.00 0.00 - yes Open
2151 5.195975268662219 -1.34677 -33.3538 9 12 0 0.00 0.00 - yes Open
2159 5.40268606994125 -1.29394 -35.4595 11 12 0 0.00 0.00 - yes Open
2309 5.477613354378612 -1.03386 -26.0639 6 18 0 0.00 0.00 - yes Open
2852 5.763934587842371 -0.866719 -22.7731 12 13 0 0.00 0.00 - yes Open
2315 5.979751350531798 -0.884627 -22.3851 7 15 0 0.00 0.00 - yes Open
2150 6.131784139044379 -1.24027 -29.2668 7 14 0 0.00 0.00 - yes Open
2698 6.149446255315745 -0.83098 -16.2148 7 13 0 0.00 0.00 - yes Open
2699 6.164468345883977 -0.769068 -20.0701 6 8 0 0.00 0.00 - yes Open
2308 6.253153426214822 -1.02266 -22.0713 9 16 0 0.00 0.00 - yes Open
2313 6.32676712506526 -0.895484 -25.3707 4 15 0 0.00 0.00 - yes Open
2312 6.46196982380152 -1.04999 -26.7339 15 14 0 0.00 0.00 - yes Open
2851 6.488641715437596 -0.92096 -22.0458 11 15 0 0.00 0.00 - yes Open
2157 6.538367177117299 -1.16091 -27.1125 9 10 0 0.00 0.00 - yes Open
2257 6.5516031034154665 -1.05698 -23.3432 6 19 0 0.00 0.00 - yes Open
2692 6.644502878033865 -0.959593 -23.3189 11 13 0 0.00 0.00 - yes Open
2256 6.680921284901709 -0.903 -21.0665 7 12 0 0.00 0.00 - yes Open
2304 6.74018410209604 -1.0249 -25.1927 15 16 0 0.00 0.00 - yes Open
2694 6.881891542076934 -0.883578 -19.5865 12 12 0 0.00 0.00 - yes Open
1698 6.978943285099711 -0.809757 -19.7782 2 16 11 0.52 0.00 - yes Current
2261 6.981018977518304 -0.792255 -17.5074 7 11 0 0.00 0.00 - yes Open
2703 6.995927191212025 -0.661673 -17.0396 6 11 0 0.00 0.00 - yes Open
2858 7.038083433074646 -0.920466 -22.9527 8 15 0 0.00 0.00 - yes Open
2855 7.078355801420884 -0.881968 -21.8367 10 15 0 0.00 0.00 - yes Open
1695 7.127794819314914 -0.916337 -18.5209 1 15 13 0.62 0.00 - yes Open
2154 7.310304338966226 -1.22813 -30.2025 6 17 0 0.00 0.00 - yes Open
1697 7.352398777778258 -0.861217 -18.4317 5 16 14 0.67 0.00 - yes Open
2258 7.417414384316499 -0.904906 -23.6753 4 14 0 0.00 0.00 - yes Open
2696 7.584661773215487 -0.843895 -17.9195 11 12 0 0.00 0.00 - yes Open
2857 7.743810824877735 -0.806387 -22.4972 6 13 0 0.00 0.00 - yes Open
2307 7.834922109443684 -1.00004 -23.4627 8 17 0 0.00 0.00 - yes Open
2314 7.971473461198626 -1.02376 -26.8634 10 14 0 0.00 0.00 - yes Open
2853 8.074202097217492 -0.991814 -24.7565 11 13 0 0.00 0.00 - yes Open
2155 8.164723108494345 -1.31131 -28.3773 11 12 0 0.00 0.00 - yes Open
2264 8.277005922310831 -0.777174 -19.5024 4 13 0 0.00 0.00 - yes Open
2849 8.283082621764063 -0.969465 -22.2867 12 16 0 0.00 0.00 - yes Open
2152 8.351732031733214 -1.13325 -23.3181 6 20 0 0.00 0.00 - yes Open
2265 8.43094888666997 -0.862862 -22.3796 4 19 0 0.00 0.00 - yes Open
2856 8.434280091431093 -0.937641 -18.4193 7 15 0 0.00 0.00 - yes Open
2693 8.575683290247046 -0.809478 -18.0789 5 10 0 0.00 0.00 - yes Open
2695 8.60181508740786 -0.703152 -18.86 4 7 0 0.00 0.00 - yes Open
2306 8.639403580829127 -1.0718 -26.3483 8 13 0 0.00 0.00 - yes Open
2260 8.853529583101354 -0.943679 -23.8904 7 12 0 0.00 0.00 - yes Open
2854 8.88911229689764 -1.08342 -24.739 13 17 0 0.00 0.00 - yes Open
2702 9.540798408787307 -0.711734 -16.7331 10 11 0 0.00 0.00 - yes Open
2700 9.721043821260514 -0.728871 -17.9387 6 9 0 0.00 0.00 - yes Open
2701 10.668134058355779 -0.712771 -20.9607 7 7 0 0.00 0.00 - yes Open
2153 14.599240275093354 -1.35261 -34.5795 9 20 0 0.00 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -19.778kcal/mol
Ligand efficiency (LE) -0.7911kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -7.192
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 25HA

Physicochemical properties

Molecular weight 356.4Da
Lipinski: ≤ 500 Da
LogP (cLogP) 2.23
Lipinski: ≤ 5
Rotatable bonds 5

Conformational strain (MMFF94s)

Strain energy (ΔE) 17.07kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 73.05kcal/mol
Minimised FF energy 55.97kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.